SCHEMBL8779192

SCHEMBL8779192

C[C@H](N)C(=O)NC(=O)Oc1nccc(OCc2ccc(Cl)cc2)c1O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CYP3A4 P08684 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
NFKB1 P19838 1/20 0.37
CYP2C19 P33261 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
MMP2 P08253 1/20 0.37
CA9 Q16790 1/20 0.37
LMNA P02545 1/20 0.37
PMP22 Q01453 1/20 0.37
NLRP3 Q96P20 1/20 0.37
INPPL1 O15357 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779134 0.91 CARM1 (0.38) KDM4EL3MBTL1ALDH1A1MMP2LMNA
SCHEMBL8779153 0.90 CARM1 (0.40) KDM4EL3MBTL1MEN1ALDH1A1KMT2A
SCHEMBL8779198 0.89 LTA4H (0.46) KDM4EL3MBTL1ALDH1A1SMN1; SMN2CYP2C9
SCHEMBL8779316 0.88 MME (0.39) KDM5APPARGMAOB
SCHEMBL8779265 0.85 TRPV1 (0.38) MMP2PPARGLTA4HMRGPRX4
SCHEMBL8779168 0.84 SMN1; SMN2 (0.40) L3MBTL1MEN1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL8779212 0.83 HPGD (0.38) KDM4EL3MBTL1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL8779176 0.83 HPGD (0.38) KDM4EL3MBTL1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL8882950 0.83 KMT2A (0.41) KDM4EL3MBTL1MEN1ALDH1A1KMT2A
SCHEMBL8779292 0.82 CARM1 (0.35) SMN1; SMN2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed