SCHEMBL8779264

SCHEMBL8779264

COc1ccnc(OC(=O)NC(=O)[C@H](C)N)c1O

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 7/20 0.35
CARM1 Q86X55 3/20 0.34
PRMT6 Q96LA8 3/20 0.34
GRIN3B O60391 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2C Q14957 1/20 0.33
IKBKB O14920 1/20 0.32
CIT O14578 2/20 0.32
ALDH1A1 P00352 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CYP3A4 P08684 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779308 0.89 ALDH1A1 (0.36) CARM1PRMT6GRIN3BGRIN1GRIN2C
SCHEMBL8779267 0.89 ALDH1A1 (0.36) CARM1PRMT6GRIN3BGRIN1GRIN2C
SCHEMBL8779212 0.88 HPGD (0.38) AAK1CARM1PRMT6GRIN3BGRIN1
SCHEMBL8779176 0.88 HPGD (0.38) AAK1CARM1PRMT6GRIN3BGRIN1
SCHEMBL8779292 0.86 CARM1 (0.35) AAK1CARM1PRMT6CYP3A4
SCHEMBL8779183 0.86 REN (0.35) CARM1PRMT6IKBKB
SCHEMBL8779140 0.86 REN (0.35) CARM1PRMT6IKBKB
SCHEMBL8779325 0.85 IKBKB (0.37) CARM1PRMT6IKBKBALDH1A1LMNA
SCHEMBL8779136 0.85 IKBKB (0.37) CARM1PRMT6IKBKBALDH1A1LMNA
SCHEMBL8779135 0.84 XIAP (0.40) CARM1PRMT6CYP3A4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed