SCHEMBL8779925

SCHEMBL8779925

O=C(N[C@H](CC(=O)c1nc2ccccc2[nH]1)C(=O)OCc1ccccc1)OCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.48
HDAC4 P56524 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC10 Q969S8 1/20 0.48
HDAC11 Q96DB2 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
HDAC9 Q9UKV0 1/20 0.48
HDAC5 Q9UQL6 1/20 0.48
DAGLA Q9Y4D2 1/20 0.48
ITGB3 P05106 10/20 0.47
ITGAV P06756 10/20 0.47
ITGA2B P08514 2/20 0.45
ITGB5 P18084 1/20 0.45
IDO1 P14902 1/20 0.44
NOS1 P29475 1/20 0.44
AAK1 Q2M2I8 1/20 0.44
CASP1 P29466 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779881 1.00 HDAC3 (0.48) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL9687293 0.87 EGLN1 (0.43) IDO1NOS1AAK1CASP1
SCHEMBL8779934 0.87 AAK1 (0.45) ITGB3ITGAVIDO1NOS1AAK1
SCHEMBL6528186 0.76 PIN1 (0.59) ITGB3ITGAVITGA2B
SCHEMBL21240753 0.76 DAGLA (0.54) DAGLAFAAH
SCHEMBL7419324 0.76 CASP1 (0.54) IDO1CASP1
SCHEMBL7419321 0.76 CASP1 (0.54) IDO1CASP1
SCHEMBL9516878 0.76 PADI4 (0.51) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL4280674 0.76 CASP1 (0.67) CASP1
SCHEMBL4280669 0.76 CASP1 (0.67) CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0539057-B1 Benzimidazole phosphono-amino acids AMERICAN HOME PROD (US) 1997-07-16 EP disclosed
EP-0539057-A1 Benzimidazole phosphono-amino acids AMERICAN HOME PRODUCTS CORPORATION (US) 1993-04-28 EP disclosed
US-5124319-A Administering for treatment of neuropathological disorders induced by overstimulation of excitatory amino acid receptors AMERICAN HOME PRODUCTS CORPORATION (US) 1992-06-23 US disclosed