SCHEMBL8780486

SCHEMBL8780486

CCC(C)c1cc2ccccc2c(Cc2ccc(C(=O)O)cc2)n1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.39
PDE7A Q13946 1/20 0.39
PDE7B Q9NP56 1/20 0.39
SRD5A2 P31213 2/20 0.38
TSHR P16473 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 2/20 0.38
DHFR P00374 1/20 0.37
TSPO P30536 1/20 0.36
RARG P13631 1/20 0.35
RORC P51449 1/20 0.35
APOBEC3A P31941 1/20 0.35
APOBEC3G Q9HC16 1/20 0.35
EGFR P00533 1/20 0.35
KDR P35968 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9119211 0.76 RARB (0.47) ALDH1A1LMNA
SCHEMBL7838471 0.74 RXRA (0.49) ALDH1A1LMNA
SCHEMBL7849442 0.72 RXRA (0.43) PDE7APDE7B
SCHEMBL7839571 0.71 SMN1; SMN2 (0.43) SRD5A2ALDH1A1LMNA
SCHEMBL8780435 0.70 TSHR (0.45) NR1H4PDE7APDE7BSRD5A2TSHR
SCHEMBL8780448 0.68 PDE7A (0.45) PDE7APDE7BALDH1A1LMNADHFR
SCHEMBL12126296 0.67 PTPN1 (0.55) TSHRALDH1A1
SCHEMBL4058443 0.66 ADAM17 (0.54) PDE7APDE7BSRD5A2TSHRALDH1A1
SCHEMBL30977564 0.65 LTB4R (0.43) ALDH1A1LMNAAPOBEC3AAPOBEC3G
SCHEMBL1682210 0.65 LTB4R (0.43) ALDH1A1LMNAAPOBEC3AAPOBEC3G

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0498722-B1 Bicyclic nitrogen compounds, their preparation, intermediates obtained, their use as pharmaceuticals and pharmaceutical compositions containing them ROUSSEL UCLAF (FR) 1997-07-30 EP disclosed
EP-0498722-A1 Bicyclic nitrogen compounds, their preparation, intermediates obtained, their use as pharmaceuticals and pharmaceutical compositions containing them ROUSSEL UCLAF (FR) 1992-08-12 EP disclosed