SCHEMBL8780947

SCHEMBL8780947

CCCN(CCCc1cc(=O)n(C)c(=O)n1C)CCc1ccccc1N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.39
SIGMAR1 Q99720 1/20 0.36
DRD2 P14416 3/20 0.35
CYP3A4 P08684 2/20 0.35
KCNH2 Q12809 2/20 0.35
KDM4E B2RXH2 2/20 0.35
LMNA P02545 1/20 0.35
CHRM2 P08172 1/20 0.35
ADRA2A P08913 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
ADRA2B P18089 1/20 0.35
DRD1 P21728 1/20 0.35
DRD4 P21917 1/20 0.35
DRD5 P21918 1/20 0.35
HTR2A P28223 1/20 0.35
MAPK1 P28482 1/20 0.35
CYP2C19 P33261 1/20 0.35
ADRA1A P35348 1/20 0.35
HRH1 P35367 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8780790 0.84 BCHE (0.42) HTR1ASIGMAR1KCNH2LMNAKMT2A
SCHEMBL8780889 0.82 SLC22A2 (0.40) SIGMAR1DRD2CYP3A4KCNH2KDM4E
SCHEMBL8780974 0.81 DRD2 (0.42) SIGMAR1DRD2CYP3A4KDM4ECYP2D6
SCHEMBL8780859 0.81 SLC22A2 (0.42) KCNH2GPR84SLC22A2ADRB1SLC6A4
SCHEMBL8780897 0.78 SLC22A2 (0.46) KCNH2KDM4EMAPK1RAB9AHSD17B10
SCHEMBL8780752 0.77 MAPT (0.45) HTR1ASIGMAR1DRD2CYP3A4KCNH2
SCHEMBL8780776 0.77 MAOA (0.37) HTR1ACYP3A4KCNH2LMNACHRM2
SCHEMBL8780893 0.74 KCNH2 (0.59) HTR1AKCNH2KDM4ELMNACHRM2
SCHEMBL8781005 0.74 KCNH2 (0.57) SIGMAR1CYP3A4KCNH2SMN1; SMN2SLC22A2
SCHEMBL8780744 0.74 SLC22A2 (0.48) SIGMAR1DRD2KCNH2LMNACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0697407-B1 Pyrimidinedione derivatives and antiarrhythmic compositions containing same MITSUI TOATSU CHEMICALS (JP) 1997-06-25 EP disclosed
EP-0697407-A1 Pyrimidinedione derivatives and antiarrhythmic compositions containing same MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-02-21 EP disclosed