SCHEMBL878150

SCHEMBL878150

CS(=O)(=O)NC(Cl)(CCC(=O)O)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.38
HIF1A Q16665 1/20 0.38
ALDH1A1 P00352 2/20 0.37
ESR1 P03372 1/20 0.37
CYP3A4 P08684 1/20 0.37
ESR2 Q92731 1/20 0.37
CYP1A2 P05177 1/20 0.37
NR3C2 P08235 1/20 0.36
CYP2D6 P10635 1/20 0.36
MAPK1 P28482 1/20 0.36
KCNN4 O15554 1/20 0.34
TBXA2R P21731 1/20 0.34
KEAP1 Q14145 2/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC11 Q96DB2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2364654 0.78 CYP2C19 (0.40) CYP2C19HIF1AALDH1A1ESR1CYP3A4
SCHEMBL877681 0.78 CYP2C19 (0.37) CYP2C19HIF1AALDH1A1ESR1CYP3A4
SCHEMBL27621428 0.71 CYP1A2 (0.48) CYP2C19HIF1AALDH1A1ESR1CYP3A4
SCHEMBL877144 0.70 MMP12 (0.38) HIF1AALDH1A1ESR1CYP3A4ESR2
SCHEMBL28021844 0.70 CYP1A2 (0.47) CYP2C19HIF1AALDH1A1ESR1CYP3A4
SCHEMBL27679367 0.68 CYP2C19 (0.50) CYP2C19HIF1AALDH1A1CYP3A4CYP1A2
SCHEMBL27942173 0.68 ALDH1A1 (0.39) CYP2C19HIF1AALDH1A1ESR1CYP1A2
SCHEMBL27623245 0.68 HDAC3 (0.40) CYP2C19HIF1ACYP1A2CYP2D6MAPK1
SCHEMBL1682512 0.68 HIF1A (0.53) CYP2C19HIF1AALDH1A1ESR1CYP3A4
SCHEMBL75391 0.68 ALDH1A1 (0.72) CYP2C19HIF1AALDH1A1ESR1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619179-A1 MATRIX METALLOPROTEINASE INHIBITORS Ranbaxy Laboratories Limited (IN) 2013-07-31 EP claimed
WO-2012038944-A1 MATRIX METALLOPROTEINASE INHIBITORS RANBAXY LABORATORIES LIMITED (IN) 2012-03-29 WO claimed