SCHEMBL8784254

SCHEMBL8784254

CNCC(c1ccccc1)N1CCC(N2CCCCC2)CC1

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
L3MBTL3 Q96JM7 2/20 0.58
L3MBTL1 Q9Y468 1/20 0.58
TACR1 P25103 4/20 0.54
CCR3 P51677 12/20 0.50
MBTD1 Q05BQ5 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
TSHR P16473 1/20 0.46
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16333179 0.84 CYP1A2 (0.57) CCR3CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL7727307 0.84 CYP1A2 (0.57) CCR3CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL6478479 0.84 CYP1A2 (0.57) CCR3CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL20246717 0.81 SIGMAR1 (0.47) CCR3CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL8784212 0.81 TACR1 (0.64) TACR1CYP3A4CYP2D6CYP2C19
SCHEMBL4070780 0.76 HRH3 (0.50) CCR3CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL1461270 0.75 MC4R (0.53) L3MBTL3L3MBTL1TACR1CCR3MBTD1
SCHEMBL11968795 0.75 MC4R (0.57) L3MBTL3L3MBTL1TACR1CCR3TSHR
SCHEMBL23682663 0.75 L3MBTL3 (1.00) L3MBTL3L3MBTL1MBTD1CYP2D6CYP2C19
SCHEMBL8276876 0.74 ALDH1A1 (0.49) CCR3CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0781277-A1 NEUROKININ ANTAGONISTS BOEHRINGER INGELHEIM KG (DE) 1997-07-02 EP disclosed
WO-1996008480-A1 NEUROKININ ANTAGONISTS BOEHRINGER INGELHEIM KG (DE) 1996-03-21 WO disclosed