SCHEMBL7727307

SCHEMBL7727307

CNC[C@@H](c1ccccc1)N1CCCC1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 6/20 0.57
CYP2C19 P33261 6/20 0.57
CYP3A4 P08684 5/20 0.57
CYP2D6 P10635 5/20 0.57
TSHR P16473 1/20 0.57
CYP2C9 P11712 5/20 0.50
KCNA5 P22460 4/20 0.50
KCNH2 Q12809 4/20 0.50
HPGD P15428 1/20 0.50
MAPK1 P28482 1/20 0.50
CCR3 P51677 2/20 0.49
KCNE1 P15382 1/20 0.48
ALDH1A1 P00352 2/20 0.48
TAAR1 Q96RJ0 1/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
SLC6A3 Q01959 2/20 0.44
MC4R P32245 1/20 0.43
GLA P06280 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16333179 1.00 CYP1A2 (0.57) CYP1A2CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL6478479 1.00 CYP1A2 (0.57) CYP1A2CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL4070780 0.90 HRH3 (0.50) CYP1A2CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL8276876 0.85 ALDH1A1 (0.49) CYP2C19CYP3A4CYP2C9KCNA5MAPK1
SCHEMBL14438305 0.84 CYP1A2 (0.56) CYP1A2CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL8784254 0.84 L3MBTL3 (0.58) CYP1A2CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL20246717 0.83 SIGMAR1 (0.47) CYP1A2CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL4061635 0.83 MAPT (0.43) CYP1A2CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL18664522 0.82 CYP1A2 (0.57) CYP1A2CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL4063476 0.81 MBTD1 (0.46) CYP1A2CYP2C19CYP3A4CYP2D6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6391910-B1 OPIOID ANTAGONIST; ANALGESIC ADOLOR CORPORATION 2002-05-21 US disclosed