SCHEMBL8787679

SCHEMBL8787679

CCCCCN1CCN(CCCCc2ccc3c(c2)OCC(=O)N3)CC1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 10/20 0.53
HTR1A P08908 10/20 0.53
HTR2A P28223 3/20 0.53
HTR1D P28221 7/20 0.53
HTR1B P28222 7/20 0.53
DRD4 P21917 9/20 0.53
DRD3 P35462 9/20 0.53
SLC6A4 P31645 5/20 0.52
KCNH2 Q12809 2/20 0.52
SIGMAR1 Q99720 2/20 0.50
CHRM5 P08912 1/20 0.50
ADRA2A P08913 1/20 0.50
ADRA2B P18089 1/20 0.50
ADRA1B P35368 1/20 0.50
TMEM97 Q5BJF2 1/20 0.50
PARP1 P09874 1/20 0.48
HTR2C P28335 1/20 0.44
HTR2B P41595 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9594420 0.84 DRD4 (0.74) DRD2HTR1AHTR2AHTR1DHTR1B
SCHEMBL8786686 0.83 DRD2 (0.60) DRD2HTR1AHTR2AHTR1DHTR1B
SCHEMBL8195715 0.82 PARP1 (0.60) DRD2HTR1AHTR2AHTR1DHTR1B
SCHEMBL8785358 0.81 HTR1A (0.73) DRD2HTR1AHTR2AHTR1DHTR1B
SCHEMBL14510673 0.80 HTR1A (0.62) DRD2HTR1AHTR2AHTR1DHTR1B
SCHEMBL9595103 0.78 HTR1A (0.71) DRD2HTR1AHTR2ADRD4DRD3
SCHEMBL9449665 0.78 MAOB (0.48) DRD2HTR1AHTR2ADRD4DRD3
SCHEMBL21207261 0.77 PARP1 (0.74) DRD2HTR1AHTR1DHTR1BDRD4
SCHEMBL12346687 0.77 HTR1A (0.58) DRD2HTR1AHTR2AHTR1DHTR1B
SCHEMBL2056366 0.77 PARP1 (0.77) DRD2HTR1AHTR2ADRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0478446-B1 Heterocyclic alkylamines, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 1997-11-19 EP claimed
EP-0478446-A1 Heterocyclic alkylamines, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1992-04-01 EP claimed