SCHEMBL8795255

SCHEMBL8795255

CCOC(=O)c1[nH]c2cc(C(F)(F)F)ccc2c1C(=O)OCC

nearest known ligand 0.69

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 13/20 0.57
MAPT P10636 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19831095 0.88 ALOX15 (0.53) ALOX15
SCHEMBL8540507 0.86 KDM4E (0.60) ALOX15MAPT
SCHEMBL29777 0.82 MAPT (0.48) MAPT
SCHEMBL15622226 0.82 HTR6 (0.50) ALOX15MAPT
SCHEMBL4126314 0.82 ALDH1A1 (0.58) MAPT
SCHEMBL31486199 0.81 ALOX5 (0.46) ALOX15MAPT
SCHEMBL15622314 0.81 HTR6 (0.49) ALOX15MAPT
SCHEMBL31423315 0.81 ALDH1A1 (0.46) MAPT
SCHEMBL8793660 0.80 ALOX15 (0.85) ALOX15
SCHEMBL8795754 0.80 ALOX15 (0.61) ALOX15MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5652239-A TREATMENT OF STROKES, ISCHEMIC ATTACK, ANTAGONISTS OF EXCITATORY AMINO ACIDS GLUTAMATE AND ASPARTATE IMPERIAL CHEMICAL COMPANY (GB) 1997-07-29 US disclosed
EP-0512817-B1 Pyridazinedione derivatives, their preparation and pharmaceutical applications ZENECA LTD (GB) 1997-02-19 EP disclosed
EP-0512817-A1 Pyridazinedione derivatives, their preparation and pharmaceutical applications ZENECA LIMITED (GB) 1992-11-11 EP disclosed