SCHEMBL8795261

SCHEMBL8795261

CCC(C)(C)c1ccc(OCC(=O)Nc2c[c]ccc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MDH1 P40925 3/20 0.51
MDH2 P40926 3/20 0.51
HIF1A Q16665 1/20 0.50
EPAS1 Q99814 1/20 0.50
MLYCD O95822 1/20 0.46
HPGD P15428 1/20 0.45
TRPV1 Q8NER1 2/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
MAPT P10636 2/20 0.44
ALDH1A1 P00352 2/20 0.44
MAPK1 P28482 1/20 0.44
KDM4E B2RXH2 1/20 0.44
HCAR2 Q8TDS4 1/20 0.44
LMNA P02545 1/20 0.43
POLB P06746 1/20 0.43
TP53 P04637 1/20 0.43
NPC1 O15118 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15467807 0.85 MDH1 (0.60) MDH1MDH2HIF1AEPAS1MLYCD
SCHEMBL7208905 0.84 NPSR1 (0.55) MDH1MDH2HIF1AEPAS1TRPV1
SCHEMBL6332042 0.81 LMNA (0.58) MLYCDHPGDSMN1; SMN2MAPTALDH1A1
SCHEMBL31303632 0.78 HIF1A (0.81) MDH1MDH2HIF1AEPAS1SMN1; SMN2
SCHEMBL2957387 0.78 HIF1A (0.81) MDH1MDH2HIF1AEPAS1SMN1; SMN2
SCHEMBL5263982 0.74 KMT2A (0.58) HPGDSMN1; SMN2ALDH1A1MAPK1KDM4E
SCHEMBL1419452 0.74 HPGD (0.58) HPGDSMN1; SMN2MAPTALDH1A1MAPK1
SCHEMBL359542 0.72 GAA (0.54) HPGDSMN1; SMN2MAPTALDH1A1MAPK1
SCHEMBL11088061 0.71 RAB9A (0.58) HPGDSMN1; SMN2MAPTALDH1A1KDM4E
SCHEMBL31503974 0.71 TRPV1 (0.70) MDH1MDH2HIF1AEPAS1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0755394-A1 A METHOD OF INDUCING CHOLECYSTOKININ AGONIST ACTIVITY USING 1,4-BENZODIAZEPINE COMPOUNDS GLAXO WELLCOME INC. (US) 1997-01-29 EP disclosed
WO-1995028399-A1 A METHOD OF INDUCING CHOLECYSTOKININ AGONIST ACTIVITY USING 1,4-BENZODIAZEPINE COMPOUNDS GLAXO WELLCOME INC. (US) 1995-10-26 WO disclosed