SCHEMBL8797294

SCHEMBL8797294

CCc1cccc(CC)c1NC(=O)OC1c2ccccc2COc2cc(C)c(Br)c(C)c21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.38
NLRP3 Q96P20 2/20 0.36
MAPT P10636 5/20 0.36
ALDH1A1 P00352 2/20 0.36
TDP1 Q9NUW8 3/20 0.34
ROCK2 O75116 1/20 0.33
HTT P42858 2/20 0.32
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
GLA P06280 1/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
RAB9A P51151 1/20 0.32
ATM Q13315 1/20 0.32
THRB P10828 1/20 0.32
LMNA P02545 1/20 0.32
POLB P06746 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8797278 0.87 TP53 (0.41) TP53NLRP3MAPTALDH1A1TDP1
SCHEMBL8797254 0.86 NLRP3 (0.36) TP53NLRP3MAPTALDH1A1LMNA
SCHEMBL8797616 0.82 TP53 (0.39) TP53NLRP3MAPTTDP1ROCK2
SCHEMBL8797282 0.77 TP53 (0.44) TP53MAPTALDH1A1HTTRAB9A
SCHEMBL8797337 0.75 ALDH1A1 (0.42) MAPTALDH1A1TBXA2R
SCHEMBL8797543 0.74 TP53 (0.39) TP53NLRP3MAPTALDH1A1TDP1
SCHEMBL8798136 0.72 TP53 (0.42) TP53NLRP3ALDH1A1LMNAKMT2A
SCHEMBL8798200 0.72 TP53 (0.48) TP53MAPTTDP1ROCK2HTT
SCHEMBL8620574 0.71 TBXA2R (0.40) MAPTALDH1A1TBXA2R
SCHEMBL8797534 0.71 NLRP3 (0.39) TP53NLRP3ALDH1A1TDP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0497201-B1 Tricyclic compounds and intermediates thereof KYOWA HAKKO KOGYO KK (JP) 1997-01-15 EP claimed