SCHEMBL8798677

SCHEMBL8798677

Nc1ccc(N)c([N+](=O)[O-])c1CC(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
USP2 O75604 1/20 0.39
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39
TDP1 Q9NUW8 5/20 0.39
CYP3A4 P08684 2/20 0.39
ALOX15 P16050 1/20 0.39
MAPT P10636 3/20 0.35
TSHR P16473 2/20 0.35
POLB P06746 1/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA5A P35218 1/20 0.34
CA9 Q16790 1/20 0.34
GAA P10253 1/20 0.33
THRB P10828 1/20 0.33
PDE7A Q13946 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8797902 0.79 ALDH1A1 (0.43) ALDH1A1KMT2ATDP1MAPTTSHR
SCHEMBL8798720 0.78 ALDH1A1 (0.46) ALDH1A1MEN1KMT2ACYP3A4MAPT
SCHEMBL77335 0.76 POLB (0.46) ALDH1A1MEN1KMT2AUSP2KEAP1
SCHEMBL8799644 0.75 GLA (0.38) ALDH1A1MEN1KMT2AMAPTPOLB
SCHEMBL8797956 0.74 ADRB2 (0.32) ALDH1A1
SCHEMBL27832802 0.73 MEN1 (0.53) ALDH1A1MEN1KMT2AUSP2KEAP1
SCHEMBL1933923 0.73 TSHR (0.47) ALDH1A1MEN1KMT2AUSP2KEAP1
SCHEMBL19952852 0.71 IMPDH2 (0.41) ALDH1A1MEN1KMT2AUSP2KEAP1
SCHEMBL14638102 0.71 HTT (0.44) ALDH1A1MEN1KMT2AUSP2KEAP1
SCHEMBL4365843 0.70 POLB (0.48) ALDH1A1MEN1KMT2AUSP2KEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0532039-B1 N1-trifluoroalkyl substituted 2-nitro-p-phenylenediamine dyes BRISTOL MYERS SQUIBB CO (US) 1997-12-03 EP claimed
EP-0532039-A1 N1-trifluoroalkyl substituted 2-nitro-p-phenylenediamine dyes Bristol-Myers Squibb Company (US) 1993-03-17 EP claimed
EP-0532039-B1 N1-trifluoroalkyl substituted 2-nitro-p-phenylenediamine dyes BRISTOL MYERS SQUIBB CO (US) 1997-12-03 EP disclosed
EP-0532039-A1 N1-trifluoroalkyl substituted 2-nitro-p-phenylenediamine dyes Bristol-Myers Squibb Company (US) 1993-03-17 EP disclosed