SCHEMBL8799334

SCHEMBL8799334

O=C(c1ccc(OCc2cscn2)cc1CC1CCCCC1)c1ccc(OCc2cscn2)cc1CC1CCCCC1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.46
MET P08581 1/20 0.40
PARP10 Q53GL7 4/20 0.38
PKM P14618 1/20 0.38
PARP15 Q460N3 3/20 0.37
CACNA1B Q00975 1/20 0.36
MAOB P27338 5/20 0.34
ACHE P22303 1/20 0.34
ALOX5AP P20292 2/20 0.34
MMP2 P08253 1/20 0.34
MMP9 P14780 1/20 0.34
MAOA P21397 1/20 0.33
MMP13 P45452 1/20 0.33
MMP14 P50281 1/20 0.33
P2RX1 P51575 1/20 0.33
S1PR1 P21453 1/20 0.33
SCN9A Q15858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8799338 0.76 ALOX5 (0.52) ALOX5PARP10PARP15CACNA1BMMP13
SCHEMBL8800932 0.71 ALOX5 (0.46) ALOX5CACNA1BMMP13MMP14
SCHEMBL8799902 0.70 ALOX5 (0.53) ALOX5CACNA1BMMP13MMP14
SCHEMBL17760501 0.69 SCN9A (0.37) ALOX5P2RX1SCN9A
SCHEMBL3590769 0.69 MAOB (0.46) ALOX5METPARP10PKMPARP15
SCHEMBL28168093 0.68 SLC6A3 (0.36) ALOX5P2RX1SCN9A
Lithium Ion SCHEMBL3590770 0.68 MAOB (0.42) ALOX5METPARP10PKMPARP15
SCHEMBL20305349 0.67 ALOX5 (0.39) ALOX5METMAOBMAOAMMP13
SCHEMBL8801528 0.67 ALOX5 (0.51) ALOX5CACNA1B
SCHEMBL3583451 0.67 MAOB (0.44) ALOX5METPARP10PKMMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0772594-A1 IMINOXYCARBOXYLATES AND DERIVATIVES AS INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS Abbott Laboratories (US) 1997-05-14 EP disclosed
US-5512581-A ANTIINFLAMMATORY AGENT ABBOTT LABORATORIES (US) 1996-04-30 US disclosed
WO-1996002507-A1 IMINOXYCARBOXYLATES AND DERIVATIVES AS INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS ABBOTT LABORATORIES (US) 1996-02-01 WO disclosed