SCHEMBL8799363

SCHEMBL8799363

Fc1cccc2c1OC(Br)C2Br

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.35
HTR2B P41595 2/20 0.35
ADRA2A P08913 1/20 0.31
KDM1A O60341 2/20 0.31
TERT O14746 1/20 0.31
KDM1B Q8NB78 1/20 0.31
CHRNB2 P17787 1/20 0.30
CHRNA4 P43681 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29363771 0.76 HTR2A (0.36) HTR2CHTR2BADRA2A
SCHEMBL18536296 0.68 MEN1 (0.37) HTR2CHTR2BADRA2AKDM1ATERT
SCHEMBL3370754 0.66 MAOA (0.38)
SCHEMBL6417599 0.66 MAOA (0.38)
SCHEMBL3370745 0.66 MAOA (0.38)
SCHEMBL3370749 0.66 MAOA (0.38)
SCHEMBL30499165 0.65 CA2 (0.41) TERT
SCHEMBL18469494 0.63 MEN1 (0.33) HTR2CHTR2BTERT
SCHEMBL25309741 0.63 HTR2C (0.36) HTR2CHTR2BCHRNB2CHRNA4
SCHEMBL30026895 0.61 CHRNB2 (0.38) HTR2CHTR2BADRA2AKDM1AKDM1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0355827-B1 Hydantoin derivatives MOCHIDA PHARM CO LTD (JP) 1997-01-02 EP disclosed
US-RE35279-E ALDOSE REDUCTASE INHIBITORS MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1996-06-18 US disclosed
US-5202339-A Hypoglycemic, hypolipedemic agents MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1993-04-13 US disclosed
US-5004751-A Antidiabetic agents; aldoe reductase inhibitors MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1991-04-02 US disclosed
WO-1990002126-A1 HYDANTOIN DERIVATIVES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1990-03-08 WO disclosed
EP-0355827-A2 Hydantoin derivatives MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1990-02-28 EP disclosed