SCHEMBL8799379

SCHEMBL8799379

C[C](C)Oc1ccc(C(C)C)cc1C#N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
IMPDH2 P12268 1/20 0.38
IMPDH1 P20839 1/20 0.38
KDM4E B2RXH2 1/20 0.38
USP2 O75604 1/20 0.38
AR P10275 3/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
ADRB2 P07550 1/20 0.35
ADRB1 P08588 1/20 0.35
ADRB3 P13945 1/20 0.35
MCL1 Q07820 1/20 0.35
XDH P47989 2/20 0.35
EGFR P00533 1/20 0.34
ERBB2 P04626 1/20 0.34
CACNA1H O95180 1/20 0.34
TRPA1 O75762 1/20 0.34
PTGS1 P23219 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL171743 0.82 MAOA (0.46) ALDH1A1IMPDH2IMPDH1KDM4EUSP2
SCHEMBL11150870 0.81 ALDH1A1 (0.58) ALDH1A1IMPDH2IMPDH1KDM4EUSP2
SCHEMBL8799381 0.79 XDH (0.48) ALDH1A1IMPDH2IMPDH1KDM4EUSP2
SCHEMBL9034189 0.77 AR (0.43) ALDH1A1IMPDH2IMPDH1KDM4EUSP2
SCHEMBL24680031 0.77 XDH (0.44) ALDH1A1ARTSHRXDHBCHE
SCHEMBL19954833 0.76 XDH (0.44) XDHACHE
SCHEMBL8799276 0.76 NOS2 (0.43) ALDH1A1KDM4EUSP2MAOAMAOB
SCHEMBL23791164 0.75 AR (0.40) ALDH1A1IMPDH2IMPDH1KDM4EUSP2
SCHEMBL17639918 0.75 ALDH1A1 (0.46) ALDH1A1ARXDHHTT
SCHEMBL9034950 0.75 NPC1 (0.51) ALDH1A1IMPDH2IMPDH1KDM4EUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0482771-B1 Heterocyclic acids ZENECA LTD (GB) 1997-06-18 EP disclosed
US-5410064-A Thromboxane A2 antagonists and inhibitors of thromboxane A2 synthase IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1995-04-25 US disclosed
US-5219874-A Heterocyclic acids IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-06-15 US disclosed
EP-0482771-A2 Heterocyclic acids ZENECA LIMITED (GB) 1992-04-29 EP disclosed