SCHEMBL8799494

SCHEMBL8799494

O=C(Nc1ccc(C(=O)N2CCCCc3sccc32)cc1)c1cccc(F)c1

nearest known ligand 0.65

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 7/20 0.65
AVPR1B P47901 4/20 0.65
AVPR2 P30518 2/20 0.63
NPC1 O15118 3/20 0.55
RAB9A P51151 3/20 0.55
SMN1; SMN2 Q16637 3/20 0.55
TP53 P04637 2/20 0.55
MAPT P10636 2/20 0.55
TSHR P16473 1/20 0.55
ALDH1A1 P00352 1/20 0.51
GLA P06280 1/20 0.51
PKM P14618 1/20 0.51
POLB P06746 1/20 0.49
KMT2A Q03164 2/20 0.48
NFKB1 P19838 1/20 0.48
HTT P42858 1/20 0.48
NFKB2 Q00653 1/20 0.48
RELA Q04206 1/20 0.48
MEN1 O00255 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6989817 0.86 AVPR1A (0.66) AVPR1AAVPR1BNPC1RAB9ASMN1; SMN2
SCHEMBL6987161 0.84 AVPR1A (0.73) AVPR1AAVPR1BAVPR2NPC1RAB9A
SCHEMBL8798138 0.83 AVPR1A (0.77) AVPR1AAVPR1BAVPR2
SCHEMBL8797050 0.83 AVPR1A (0.59) AVPR1AAVPR1BAVPR2MAPTPOLB
SCHEMBL8796877 0.82 AVPR1A (0.71) AVPR1AAVPR1BAVPR2KMT2AMEN1
SCHEMBL8797460 0.82 AVPR1A (0.62) AVPR1AAVPR1BAVPR2TP53KMT2A
SCHEMBL7365160 0.81 AVPR1A (0.68) AVPR1AAVPR1BAVPR2SMN1; SMN2TP53
SCHEMBL7348119 0.81 RAB9A (0.64) RAB9A
SCHEMBL6991783 0.79 AVPR1A (0.67) AVPR1AAVPR1BAVPR2MAPTALDH1A1
SCHEMBL6989132 0.79 AVPR1A (0.85) AVPR1AAVPR1BAVPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0811008-A1 BICYCLIC BENZAZEPINE DERIVATIVES AS VASOPRESSIN ANTAGONISTS American Cyanamid Company (US) 1997-12-10 EP disclosed