SCHEMBL8799780

SCHEMBL8799780

COC(=O)C(=O)Nc1cc(Cl)c(Oc2ccc(OC)c(C(C)C)c2)c(Cl)c1

nearest known ligand 0.78

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
RORC P51449 8/20 0.68
THRB P10828 7/20 0.68
THRA P10827 2/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22959176 0.88 RORC (0.70) RORCTHRBTHRA
SCHEMBL22959162 0.88 RORC (0.70) RORCTHRBTHRA
SCHEMBL8799735 0.87 THRA (0.67) THRBTHRA
SCHEMBL7094647 0.87 THRB (0.61) RORCTHRBTHRA
SCHEMBL7097343 0.86 THRB (0.52) RORCTHRBTHRA
SCHEMBL22959104 0.85 RORC (0.67) RORCTHRBTHRA
SCHEMBL22959193 0.84 RORC (0.74) RORCTHRBTHRA
SCHEMBL22959398 0.84 RORC (0.67) RORCTHRBTHRA
SCHEMBL22959249 0.84 RORC (0.73) RORCTHRBTHRA
SCHEMBL282518 0.84 RORC (0.64) RORCTHRBTHRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0580550-B1 Oxamic acid derivatives as hypocholesteremic agents CIBA GEIGY AG (CH) 1997-10-22 EP disclosed
US-5654468-A ANTILIPID, ANTICHOLESTEROL AGENTS CIBA-GEIGY CORPORATION (US) 1997-08-05 US disclosed
US-5569674-A ANTICHOLESTEROL AGENTS CIBA-GEIGY CORPORATION (US) 1996-10-29 US disclosed
US-5401772-A Anticholesterol agents with aromatic amines CIBA-GEIGY CORPORATION (US) 1995-03-28 US disclosed
EP-0580550-A1 Oxamic acid derivatives as hypocholesteremic agents CIBA-GEIGY AG (CH) 1994-01-26 EP disclosed