SCHEMBL8801541

SCHEMBL8801541

CCOC(=O)C(C(=O)OCC)C(=O)c1ccc(Cl)nc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
TDP1 Q9NUW8 2/20 0.37
GAA P10253 1/20 0.37
LMNA P02545 2/20 0.36
MAPT P10636 1/20 0.36
CYP1A2 P05177 1/20 0.36
DGAT1 O75907 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.35
TSHR P16473 2/20 0.35
RAB9A P51151 1/20 0.35
CASP1 P29466 1/20 0.35
KLKB1 P03952 1/20 0.34
KLK1 P06870 1/20 0.34
HTT P42858 1/20 0.34
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29550931 0.81 TSHR (0.52) ALDH1A1KDM4ETDP1MAPTCYP1A2
SCHEMBL422881 0.81 TSHR (0.52) ALDH1A1KDM4ETDP1MAPTCYP1A2
SCHEMBL492531 0.78 CYP2C19 (0.51) ALDH1A1L3MBTL1TDP1LMNACYP1A2
SCHEMBL5795930 0.78 SLC6A12 (0.36) ALDH1A1KDM4EL3MBTL1TSHRRAB9A
SCHEMBL9144675 0.77 SLC6A12 (0.37) ALDH1A1LMNAMAPTSMN1; SMN2HTT
SCHEMBL29922180 0.77 SLC6A12 (0.36) ALDH1A1KDM4EL3MBTL1GAAMAPT
SCHEMBL9686323 0.77 KEAP1 (0.51) ALDH1A1KDM4ETDP1LMNAMAPT
SCHEMBL27446237 0.76 ALDH1A1 (0.37) ALDH1A1KDM4EL3MBTL1TDP1GAA
SCHEMBL2082473 0.76 PKM (0.43) ALDH1A1KDM4ETDP1GAAMAPT
SCHEMBL29980368 0.76 PKM (0.43) ALDH1A1KDM4ETDP1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612731-B1 Novel guinolone and naphthyridone derivatives BAYER AG (DE) 1997-08-20 EP disclosed
WO-1996002540-A1 HETEROCYCLYL-1-PHENYL SUBSTITUTED QUINOLONE CARBOXYLIC ACIDS AS ANTIVIRAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1996-02-01 WO disclosed
WO-1996002539-A1 SUBSTITUTED TRIAZOLYL METHYL PHENYL NAPHTHYRIDONES BAYER AKTIENGESELLSCHAFT (DE) 1996-02-01 WO disclosed
CN-1097423-A Quinolone-and naphthyridonecarboxylic acid derivatives BAYER AG (DE) 1995-01-18 CN disclosed
EP-0612731-A1 Novel guinolone and naphthyridone derivatives BAYER AG (DE) 1994-08-31 EP disclosed
EP-0607825-A1 6-H-4-OXO-3-quinoline-carboxylic acids and their analogues as antibacterial agents BAYER AG (DE) 1994-07-27 EP disclosed