SCHEMBL880259

SCHEMBL880259

BC(=O)C1=C(C)NC(=O)CC1c1cccc2ccccc12

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.60
ALOX15 P16050 1/20 0.50
PKM P14618 1/20 0.50
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
ATM Q13315 1/20 0.49
TSHR P16473 2/20 0.48
GPBAR1 Q8TDU6 1/20 0.44
TP53 P04637 3/20 0.44
HSD17B10 Q99714 2/20 0.44
GAA P10253 1/20 0.44
MTNR1A P48039 1/20 0.44
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13522417 0.85 PKM (0.70) IDO1ALOX15PKMMEN1KMT2A
SCHEMBL14450498 0.81 IDO1 (0.56) IDO1ALOX15PKMMEN1KMT2A
SCHEMBL9387969 0.76 IDO1 (1.00) IDO1TP53HSD17B10MTNR1ALMNA
Bromide SCHEMBL28839335 0.75 IDO1 (0.97) IDO1TP53HSD17B10MTNR1ALMNA
SCHEMBL880307 0.72 IDO1 (0.70) IDO1KMT2ATP53HSD17B10MTNR1A
SCHEMBL28839376 0.71 IDO1 (0.88) IDO1ALOX15PKMTP53HSD17B10
SCHEMBL880405 0.70 HTT (0.54) PKMKMT2ATSHRGPBAR1TP53
SCHEMBL3004441 0.70 IDO1 (0.58) IDO1MEN1KMT2AATMTP53
SCHEMBL880422 0.69 MAPT (0.47) ALOX15TSHRGPBAR1TP53HSD17B10
SCHEMBL7814723 0.69 MAPT (0.53) IDO1MEN1KMT2AATMTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2433634-A2 Compounds, compositions and methods of inhibiting a-synuclein toxicity The Whitehead Institute for Biomedical Research (US) 2012-03-28 EP disclosed
EP-1802303-B1 COMPOUNDS, COMPOSITIONS AND METHODS OF INHIBITING A-SYNUCLEIN TOXICITY WHITEHEAD BIOMEDICAL INST (US) 2011-11-02 EP disclosed