SCHEMBL8803532

SCHEMBL8803532

O=C(Nc1cc(Cl)ncn1)c1ccccc1SSc1ccccc1C(=O)Nc1cc(Cl)ncn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
ALOX15 P16050 2/20 0.41
MAPK1 P28482 1/20 0.41
FGFR4 P22455 1/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
POLB P06746 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTT P42858 1/20 0.40
KDR P35968 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
EGFR P00533 1/20 0.40
ERBB3 P21860 1/20 0.40
SMO Q99835 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10172501 0.78 SMN1; SMN2 (0.57) MEN1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL8375299 0.77 CHRNB2 (0.64) MEN1KMT2ACA1CA2CA9
SCHEMBL1706080 0.74 RAB9A (0.55) RAB9A
SCHEMBL30472729 0.73 KCNMA1 (0.63) MEN1KMT2AKDR
SCHEMBL8855826 0.72 FADS1 (0.65) MEN1KMT2ACA1CA2CA9
SCHEMBL18185358 0.70 L3MBTL1 (0.48) MEN1KMT2AFGFR4NPC1EGFR
SCHEMBL8855681 0.70 CYP1A2 (0.72) CA1CA2CA9NPC1RAB9A
SCHEMBL8211768 0.70 POLB (0.47) MEN1KMT2AFGFR4SMN1; SMN2POLB
SCHEMBL10795537 0.70 FADS1 (0.68) MEN1KMT2ANPC1RAB9AHTT
SCHEMBL8855680 0.70 NPC1 (0.60) MEN1KMT2ACA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0775110-A1 ARYLTHIO COMPOUNDS AS ANTIBACTERIAL AND ANTIVIRAL AGENTS WARNER-LAMBERT COMPANY (US) 1997-05-28 EP claimed
WO-1996004242-A1 ARYLTHIO COMPOUNDS AS ANTIBACTERIAL AND ANTIVIRAL AGENTS WARNER-LAMBERT COMPANY (US) 1996-02-15 WO claimed
EP-0601486-B1 Cis-epoxide derivatives useful as irreversible HIV protease inhibitors and process and intermediates for their preparation LUCKY LTD (KR) 1997-10-29 EP disclosed
US-5668291-A THIOSUBSTITUTED PYRIDINES, TREATMENT OF AIDS AND HIV WARNER-LAMBERT COMPANY (US) 1997-09-16 US disclosed
EP-0601486-A1 Cis-epoxide derivatives useful as irreversible HIV protease inhibitors and process and intermediates for their preparation LUCKY LTD. (KR) 1994-06-15 EP disclosed