SCHEMBL8808975

SCHEMBL8808975

O=C1NC(Cc2cccc3c2ccn3Cc2ccc(C(F)(F)F)cc2C(F)(F)F)C(=O)S1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.34
PARP1 P09874 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.31
KDM1A O60341 1/20 0.30
C5AR1 P21730 1/20 0.30
ESRRA P11474 1/20 0.30
EPHX2 P34913 3/20 0.30
PPARG P37231 2/20 0.30
TRPA1 O75762 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8811090 0.89 KDM1A (0.38) KDM1AC5AR1EPHX2PPARG
SCHEMBL8811868 0.88 PARP1 (0.40) DAOPARP1PTGDR2KDM1A
SCHEMBL8809597 0.87 PARP1 (0.47) PARP1
SCHEMBL8813445 0.87 HTR6 (0.40) PARP1
SCHEMBL8810643 0.86 TACR1 (0.39) PARP1
SCHEMBL8808968 0.81 PPARG (0.41) DAOPARP1PTGDR2KDM1AC5AR1
SCHEMBL8810446 0.81 PPARG (0.38) PPARG
SCHEMBL8809697 0.80 HTR6 (0.42)
SCHEMBL8812495 0.79 TNF (0.39)
SCHEMBL8808816 0.79 HTR6 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0780389-A1 Thiazolidinedione derivatives, process for their preparation and pharmaceutical compositions containing them TOBISHI PHARMACEUTICAL CO., LTD. (JP) 1997-06-25 EP disclosed