SCHEMBL8809279

SCHEMBL8809279

N#Cc1ccccc1-c1ccc2cccc(CBr)c2n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 1/20 0.41
GRM2 Q14416 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
KCNH2 Q12809 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.35
GAA P10253 1/20 0.35
GABRG2 P18507 2/20 0.34
GABRB3 P28472 2/20 0.34
GABRA3 P34903 2/20 0.34
GABRA1 P14867 1/20 0.34
CNR2 P34972 2/20 0.34
CNR1 P21554 1/20 0.34
CTSA P10619 1/20 0.34
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
GABRA5 P31644 1/20 0.33
ESR2 Q92731 1/20 0.33
CRHR1 P34998 1/20 0.33
MET P08581 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8809434 0.78 AR (0.50) GRM2L3MBTL1GAACTSA
SCHEMBL588692 0.73 ESR2 (0.44) GABRG2GABRB3GABRA3GABRA5ESR2
SCHEMBL2575065 0.73 GABRA1 (0.39) L3MBTL1GABRG2GABRB3GABRA3GABRA1
SCHEMBL21483572 0.72 NPC1 (0.50) GRM2L3MBTL1GAAESR2
SCHEMBL8484254 0.71 KCNH2 (0.40) GRM2SLC6A2SLC6A4KCNH2L3MBTL1
SCHEMBL3644296 0.71 ESR2 (0.40) GABRG2GABRB3GABRA3CA1CA2
SCHEMBL9313614 0.71 ALDH1A1 (0.40) CNR2CA1CA2ESR2
SCHEMBL2649479 0.69 SLC6A2 (0.49) GRM2SLC6A2SLC6A4KCNH2L3MBTL1
SCHEMBL899 0.69 CYP19A1 (0.46) SLC6A2SLC6A4CA1CA2
SCHEMBL29513232 0.69 CYP19A1 (0.46) SLC6A2SLC6A4CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528762-B1 N-acyl-N-heterocyclyl- or naphthyl-alkyl amino acids as angiotensin II antagonists CIBA GEIGY AG (CH) 1997-05-07 EP disclosed
EP-0528762-A1 N-acyl-N-heterocyclyl- or naphthyl-alkyl amino acids as angiotensin II antagonists CIBA-GEIGY AG (CH) 1993-02-24 EP disclosed