SCHEMBL8812902

SCHEMBL8812902

COc1cccc(N(C(C)=O)C(C)C)c1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 12/20 0.51
MTNR1B P49286 12/20 0.51
HSD17B2 P37059 2/20 0.50
CES2 O00748 1/20 0.50
CES1 P23141 1/20 0.50
PARP1 P09874 1/20 0.47
HSD17B1 P14061 1/20 0.47
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8428661 0.82 MTNR1A (0.46) MTNR1AMTNR1BHSD17B2CES2CES1
SCHEMBL5254203 0.82 HSD17B2 (0.46) MTNR1AMTNR1BHSD17B2CES2CES1
SCHEMBL6136382 0.80 MTNR1A (0.51) MTNR1AMTNR1BHSD17B2CES2CES1
SCHEMBL26624252 0.80 MTNR1B (0.56) MTNR1AMTNR1BHSD17B2CES2CES1
SCHEMBL6511331 0.80 TRPM8 (0.52) MTNR1AMTNR1BCES2CES1PARP1
SCHEMBL11027897 0.78 HSD17B2 (0.61) MTNR1AMTNR1BHSD17B2CES2CES1
SCHEMBL1548437 0.78 MTNR1B (0.55) MTNR1AMTNR1BHSD17B2CES2CES1
SCHEMBL5897694 0.78 MTNR1A (0.44) MTNR1AMTNR1BHSD17B2
SCHEMBL27784974 0.77 ALDH1A1 (0.47) NPC1
SCHEMBL27662593 0.77 MTNR1A (0.54) MTNR1AMTNR1BHSD17B2CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0755384-A1 CCK OR GASTRIN MODULATING 1,5 BENZODIAZEPINES DERIVATIVES GLAXO WELLCOME INC. (US) 1997-01-29 EP disclosed
WO-1995028391-A1 CCK OR GASTRIN MODULATING 1,5 BENZODIAZEPINES DERIVATIVES GLAXO WELLCOME INC. (US) 1995-10-26 WO disclosed