SCHEMBL8815510

SCHEMBL8815510

CC(C)(C)Oc1ccc(C[C@H](NC(=O)O)C(=O)C=[N+]=[N-])cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 2/20 0.45
ABCB1 P08183 1/20 0.42
CTSK P43235 2/20 0.39
CTSL P07711 1/20 0.39
ITGB3 P05106 1/20 0.38
ITGA2B P08514 1/20 0.38
PLG P00747 1/20 0.38
PRSS1 P07477 1/20 0.38
PRSS2 P07478 1/20 0.38
PRSS3 P35030 1/20 0.38
ALDH1A1 P00352 1/20 0.36
PKM P14618 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
FPR2 P25090 1/20 0.36
CNR1 P21554 6/20 0.36
CNR2 P34972 5/20 0.36
PPARG P37231 2/20 0.35
CTSS P25774 1/20 0.35
KDM4E B2RXH2 1/20 0.35
KDM4A O75164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16333610 0.93 CTSK (0.44) ACACBABCB1CTSKCTSLALDH1A1
SCHEMBL3431290 0.88 ABCB1 (0.52) ACACBABCB1CTSKCTSLITGB3
SCHEMBL8814267 0.86 LDHA (0.49) ACACBFPR2
SCHEMBL8814268 0.86 LDHA (0.49) ACACBFPR2
SCHEMBL29430953 0.82 CTSL (0.58) CTSKCTSLITGB3ITGA2BCTSS
SCHEMBL18862971 0.81 ALDH1A1 (0.52) CTSLALDH1A1PKMSMN1; SMN2CTSS
SCHEMBL6927025 0.81 ALDH1A1 (0.52) CTSLALDH1A1PKMSMN1; SMN2CTSS
SCHEMBL10538691 0.81 ALDH1A1 (0.52) CTSLALDH1A1PKMSMN1; SMN2CTSS
SCHEMBL31098043 0.80 NOS2 (0.46) ACACBALDH1A1PPARG
SCHEMBL7322984 0.80 PPARG (0.55) PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5652369-A PROTEASE INHIBITOR HOFFMANN-LA ROCHE INC. (US) 1997-07-29 US disclosed
US-5620987-A Amino acid derivatives HOFFMANN-LA ROCHE INC. (US) 1997-04-15 US disclosed
US-5446161-A Protease inhibitor, viricides HOFFMANN-LA ROCHE INC. (US) 1995-08-29 US disclosed