SCHEMBL8817643

SCHEMBL8817643

COC(=O)c1cccc(-c2nc(-c3cccc(C)n3)nc3ccccc23)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 2/20 0.53
TGFBR1 P36897 6/20 0.52
ABCG2 Q9UNQ0 3/20 0.47
KDM4E B2RXH2 2/20 0.47
MAPT P10636 1/20 0.47
ABCB1 P08183 1/20 0.47
GABRG2 P18507 1/20 0.46
GABRB3 P28472 1/20 0.46
GABRA5 P31644 1/20 0.46
GABRA3 P34903 1/20 0.46
GPR84 Q9NQS5 2/20 0.45
MAPK14 Q16539 1/20 0.45
ABCC1 P33527 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.44
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.43
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
GRM5 P41594 1/20 0.43
NEK1 Q96PY6 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680584 0.82 GABRG2 (0.53) GABRG2GABRB3GABRA5GABRA3LMNA
SCHEMBL6120916 0.82 TGFBR1 (0.54) TGFBR1KDM4EMAPK14
SCHEMBL8816575 0.81 ADORA2A (0.62) PDE5AABCG2KDM4EMAPTABCB1
SCHEMBL8819255 0.81 TGFBR1 (0.47) TGFBR1ABCG2MAPTMAPK14SMN1; SMN2
SCHEMBL8814729 0.81 NR1I3 (0.54) TGFBR1ABCG2MAPTABCB1MAPK14
SCHEMBL8816445 0.79 TGFBR1 (0.46) TGFBR1MAPK14
SCHEMBL8815695 0.79 ADORA2A (0.58) TGFBR1ABCG2MAPK14
SCHEMBL8815752 0.79 MEN1 (0.51) TGFBR1KDM4EMAPTMAPK14LMNA
SCHEMBL8816177 0.79 NR1I3 (0.51) PDE5ATGFBR1ABCG2KDM4EMAPK14
SCHEMBL8817436 0.79 TGFBR1 (0.47) TGFBR1ABCG2ABCB1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012066122-A1 2 - (PYRIDIN- 2 -YL) -QUINAZOLINE DERIVATIVES AND THEIR USE AS MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-05-24 WO disclosed