SCHEMBL882483

SCHEMBL882483

CCOC(=O)c1sc(Br)nc1C(F)(F)C(F)(F)F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
HPGD P15428 3/20 0.50
CYP1A2 P05177 1/20 0.43
MAPT P10636 4/20 0.42
KDM4E B2RXH2 3/20 0.42
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
HSP90AA1 P07900 1/20 0.42
CRHBP P24387 1/20 0.42
CRHR2 Q13324 1/20 0.42
TRPM8 Q7Z2W7 3/20 0.41
POLB P06746 1/20 0.41
DHODH Q02127 3/20 0.40
LMNA P02545 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL299362 0.88 ALDH1A1 (0.52) ALDH1A1HPGDCYP1A2MAPTKDM4E
SCHEMBL10821063 0.85 ALDH1A1 (0.50) ALDH1A1HPGDCYP1A2MAPTKDM4E
SCHEMBL6266650 0.84 ALDH1A1 (0.49) ALDH1A1HPGDCYP1A2MAPTKDM4E
SCHEMBL882389 0.84 ALDH1A1 (0.72) ALDH1A1HPGDCYP1A2MAPTKDM4E
SCHEMBL2362831 0.78 ALDH1A1 (0.49) ALDH1A1HPGDCYP1A2MAPTKDM4E
SCHEMBL288785 0.76 ALDH1A1 (0.59) ALDH1A1HPGDCYP1A2MAPTKDM4E
SCHEMBL622325 0.76 ALDH1A1 (0.51) ALDH1A1HPGDCYP1A2MAPTKDM4E
SCHEMBL874267 0.76 ALDH1A1 (0.39) ALDH1A1HPGDKDM4E
SCHEMBL882714 0.76 MAPT (0.57) ALDH1A1HPGDMAPTKDM4EKMT2A
SCHEMBL2309900 0.75 ALDH1A1 (0.51) ALDH1A1HPGDCYP1A2MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038905-A1 THIENOPYRIDINE NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed
WO-2012038904-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed