SCHEMBL874267

SCHEMBL874267

O=C(O)c1sc(Br)nc1C(F)(F)C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
GPR35 Q9HC97 4/20 0.38
KDM4E B2RXH2 1/20 0.30
GAA P10253 1/20 0.30
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL873879 0.85 GPR35 (0.43) ALDH1A1HPGDTSHRGPR35SMN1; SMN2
SCHEMBL10820841 0.83 ALDH1A1 (0.53) ALDH1A1HPGDTSHRGPR35KDM4E
SCHEMBL874301 0.80 ALDH1A1 (0.40) ALDH1A1HPGDTSHRRAB9A
SCHEMBL882483 0.76 ALDH1A1 (0.50) ALDH1A1HPGDKDM4E
SCHEMBL10820886 0.73 ALDH1A1 (0.55) ALDH1A1HPGDTSHRKDM4EGAA
SCHEMBL874117 0.71 RAB9A (0.48) ALDH1A1HPGDKDM4EGAARAB9A
SCHEMBL29877075 0.70 ALDH1A1 (0.45) ALDH1A1HPGDTSHRGPR35KDM4E
SCHEMBL1778181 0.69 ALDH1A1 (0.55) ALDH1A1HPGDTSHRGPR35KDM4E
SCHEMBL625723 0.69 ALDH1A1 (0.39) ALDH1A1HPGDTSHRGPR35KDM4E
SCHEMBL874785 0.69 SMN1; SMN2 (0.41) ALDH1A1KDM4EGAARAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038905-A1 THIENOPYRIDINE NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed
WO-2012038904-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed