SCHEMBL8825418

SCHEMBL8825418

CCCCCCCCCCOc1ccc(C#Cc2ccc(C(=O)OC)cc2)nc1CCC(=O)OC

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PPARG P37231 4/20 0.41
PPARA Q07869 3/20 0.41
LTB4R Q15722 1/20 0.40
SMPD1 P17405 5/20 0.39
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
NPC1 O15118 1/20 0.37
CASP1 P29466 1/20 0.37
RAB9A P51151 1/20 0.37
THRA P10827 1/20 0.37
THRB P10828 1/20 0.37
PRKCA P17252 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8825101 0.96 MAPT (0.39) PPARGPPARALTB4RALDH1A1HPGD
SCHEMBL8825493 0.84 PPARG (0.54) PPARGPPARA
SCHEMBL8825282 0.83 LTB4R (0.54) LTB4RALDH1A1HPGD
SCHEMBL8825460 0.83 PPARG (0.43) PPARGPPARALTB4R
SCHEMBL8825193 0.82 LTB4R (0.45) PPARGPPARALTB4RNPC1PRKCA
SCHEMBL8825269 0.80 PTPN11 (0.41) ALDH1A1HPGD
SCHEMBL8825203 0.80 ALOX15 (0.36)
SCHEMBL8825152 0.78 PPARG (0.45) PPARGPPARALTB4RSMPD1THRA
SCHEMBL8825147 0.78 PPARG (0.45) PPARGPPARALTB4RSMPD1THRA
SCHEMBL8825480 0.77 LTB4R (0.46) LTB4RALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5624943-A Pyridine compounds which are useful as leukotriene-B4 -antagonists SCHERING AKTIENGESELLSCHAFT (DE) 1997-04-29 US disclosed
EP-0651745-A1 NEW PYRIDINE DERIVATIVES AS LEUKCOTRIENE B 4? ANTAGONISTS SCHERING AKTIENGESELLSCHAFT (DE) 1995-05-10 EP disclosed
WO-1994002464-A1 NEW PYRIDINE DERIVATIVES AS LEUKCOTRIENE B4 ANTAGONISTS SCHERING AKTIENGESELLSCHAFT (DE) 1994-02-03 WO disclosed