SCHEMBL8828285

SCHEMBL8828285

CN(CCCNC(=O)C/C=C/c1ccc(-n2ccnc2)cc1)CCc1ccc2c(c1)OCO2

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 17/20 0.46
NOS1 P29475 7/20 0.46
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
HPGD P15428 2/20 0.42
GAA P10253 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8828172 0.95 NOS2 (0.43) NOS2NOS1
SCHEMBL8828152 0.85 TMEM97 (0.43) GAA
SCHEMBL8828195 0.85 OPRM1 (0.44) NOS2KDM4EALDH1A1HPGDGAA
SCHEMBL9159994 0.84 MAOB (0.40) ALDH1A1
SCHEMBL8828318 0.83 DRD3 (0.44) NOS2ALDH1A1HPGDGAASMN1; SMN2
SCHEMBL8828417 0.83 L3MBTL1 (0.42) KDM4EALDH1A1GAASMN1; SMN2
SCHEMBL9156723 0.83 MAOB (0.46) KDM4EALDH1A1SMN1; SMN2
SCHEMBL8828168 0.83 DRD3 (0.45) KDM4E
SCHEMBL8828202 0.83 DRD3 (0.41) GAA
SCHEMBL9159739 0.83 MAOB (0.42) KDM4EALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607953-A ANTIISCHEMIC AGENTS EISAI CO., LTD. (JP) 1997-03-04 US disclosed
EP-0344577-B1 Butenoic or propenoic acid derivatives EISAI CO LTD (JP) 1996-10-09 EP disclosed
US-5382595-A Antiischemic agents EISAI CO., LTD. (JP) 1995-01-17 US disclosed
US-5177089-A Antiischemic agent, vasodilator EISAI CO., LTD. (JP) 1993-01-05 US disclosed
US-5047417-A Butenoic or propenoic acid derivatives EISAI CO. LTD. (JP) 1991-09-10 US disclosed
EP-0344577-A2 Butenoic or propenoic acid derivatives Eisai Co., Ltd. (JP) 1989-12-06 EP disclosed