SCHEMBL8833239

SCHEMBL8833239

C=CCOC(=O)N1C[C@@H](SC(=O)c2ccccc2)C[C@H]1CCn1cncn1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 1/20 0.36
CHRM1 P11229 1/20 0.35
CYP19A1 P11511 2/20 0.34
ALDH1A1 P00352 3/20 0.32
KDM4E B2RXH2 1/20 0.32
TP53 P04637 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
S1PR1 P21453 2/20 0.32
PTGS2 P35354 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CCR5 P51681 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9220923 1.00 ECE1 (0.36) ECE1CHRM1CYP19A1ALDH1A1KDM4E
SCHEMBL8833609 0.82 ECE1 (0.38) ECE1CHRM1CYP19A1ALDH1A1KDM4E
SCHEMBL8833657 0.81 TBXAS1 (0.40) ECE1CYP19A1ALDH1A1TP53TDP1
SCHEMBL9213848 0.81 TBXAS1 (0.40) ECE1CYP19A1ALDH1A1TP53TDP1
SCHEMBL8832778 0.81 ECE1 (0.36) ECE1CHRM1CYP19A1ALDH1A1TDP1
SCHEMBL8833096 0.80 ECE1 (0.36) ECE1CHRM1CYP19A1MEN1KMT2A
SCHEMBL8832957 0.80 ECE1 (0.36) ECE1CHRM1CYP19A1MEN1KMT2A
SCHEMBL9213699 0.80 ECE1 (0.36) ECE1CHRM1CYP19A1MEN1KMT2A
SCHEMBL8832719 0.80 ECE1 (0.34) ECE1CHRM1MEN1KMT2A
SCHEMBL8833600 0.80 LMNA (0.38) ECE1CHRM1TDP1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5608056-A Substituted 3-pyrrolidinylthio-carbapenems as antimicrobial agents FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-03-04 US disclosed
EP-0636133-A1 SUBSTITUTED 3-PYRROLIDINYLTHIO-CARBAPENEMS AS ANTIMICROBIAL AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-02-01 EP disclosed
WO-1993021186-A1 SUBSTITUTED 3-PYRROLIDINYLTHIO-CARBAPENEMS AS ANTIMICROBIAL AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-10-28 WO disclosed