SCHEMBL8835181

SCHEMBL8835181

O=C(CN1CCN(C(=O)[C@@H]2C[C@H](S)CN2C(=O)OCc2ccc([N+](=O)[O-])cc2)CC1)C(=O)OCc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 1/20 0.37
KCNH2 Q12809 1/20 0.37
MGLL Q99685 1/20 0.37
TDP1 Q9NUW8 1/20 0.36
HRH2 P25021 1/20 0.36
HRH1 P35367 1/20 0.36
NPBWR1 P48145 2/20 0.36
MCHR1 Q99705 2/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
DPP8 Q6V1X1 1/20 0.36
DPP9 Q86TI2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9042781 0.89 HRH2 (0.39) KCNJ1KCNH2HRH2HRH1NPBWR1
SCHEMBL8536750 0.88 KCNJ1 (0.42) KCNJ1KCNH2HRH2HRH1KDM4E
SCHEMBL8438589 0.88 KCNJ1 (0.42) KCNJ1KCNH2HRH2HRH1KDM4E
SCHEMBL8440367 0.88 DPP8 (0.39) KCNJ1KCNH2NPBWR1MCHR1DPP8
SCHEMBL9728223 0.88 DPP8 (0.46) TDP1NPBWR1MCHR1DPP8DPP9
SCHEMBL9040592 0.87 ALDH1A1 (0.41) TDP1HRH2HRH1NPBWR1MCHR1
SCHEMBL9040433 0.87 ALDH1A1 (0.41) TDP1HRH2HRH1NPBWR1MCHR1
SCHEMBL9119637 0.87 DPP8 (0.45) NPBWR1MCHR1ALDH1A1SMN1; SMN2DPP8
SCHEMBL8434840 0.86 HRH2 (0.41) KCNJ1KCNH2TDP1HRH2HRH1
SCHEMBL8437995 0.86 HRH2 (0.41) KCNJ1KCNH2TDP1HRH2HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5614624-A THIO SUBSTITUTED, ANTIBIOTICS, CHEMICAL INTERMEDIATES SANKYO COMPANY, LIMITED (JP) 1997-03-25 US disclosed
US-5310735-A Carbapenem derivatives having antibiotic activity, their preparation and their use SANKYO COMPANY, LIMITED (JP) 1994-05-10 US disclosed