SCHEMBL8836613

SCHEMBL8836613

NCC(=O)Nn1ccc2cc(O)ccc21

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.36
CA2 P00918 4/20 0.36
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
GAA P10253 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
GFER P55789 1/20 0.33
CYP2C9 P11712 1/20 0.32
HCAR2 Q8TDS4 1/20 0.32
CA12 O43570 1/20 0.32
CA9 Q16790 1/20 0.32
FLT3 P36888 1/20 0.32
CLK1 P49759 1/20 0.31
DYRK1A Q13627 1/20 0.31
DYRK1B Q9Y463 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
HTR2B P41595 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8836401 0.84 OXER1 (0.44) CA1CA2CA12CA9HTR2A
SCHEMBL7243122 0.80 NTSR1 (0.47) ALDH1A1KMT2ASMN1; SMN2HDAC8NTSR1
SCHEMBL8835933 0.80 HTR6 (0.44) ALDH1A1MEN1GAAKMT2ALMNA
SCHEMBL8836240 0.80 MTNR1A (0.52) ALDH1A1KDM4ESMN1; SMN2HTR2CLMNA
SCHEMBL8836533 0.80 MTNR1A (0.52) ALDH1A1KDM4ESMN1; SMN2HTR2CLMNA
SCHEMBL2870562 0.80 CA12 (0.44) CA1CA2KMT2ACA12CA9
SCHEMBL8836539 0.79 TP53 (0.43) ALDH1A1KDM4EMEN1KMT2ASMN1; SMN2
Hydrochloric Acid SCHEMBL8836099 0.78 CA12 (0.43) CA1CA2KMT2ACA12CA9
SCHEMBL8836018 0.78 AKR1C3 (0.42) ALDH1A1KDM4EKMT2ALMNA
SCHEMBL8836009 0.77 LTA4H (0.53) ALDH1A1KDM4EMEN1KMT2ACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5319096-A Neuroprotective agent HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-06-07 US claimed
US-5646300-A NEUROPROTECTIVE AGENTS HOECHST MARION ROUSSEL, INC. (US) 1997-07-08 US disclosed
US-5591866-A NEUROPROTECTIVE AGENTS HOECHST MARION ROUSSEL INC. (US) 1997-01-07 US disclosed
US-5565579-A NEUROPROTECTIVE AGENT HOECHST MARION ROUSSEL INC. (US) 1996-10-15 US disclosed
EP-0563916-B1 (1H-Indol-1-yl)-2-(amino)acetamides and related (1H-indol-1-yl)-(aminoalkyl)amides, intermediates and a process for their preparation and their use as medicaments HOECHST ROUSSEL PHARMA (US) 1995-08-16 EP disclosed
US-5319096-A Neuroprotective agent HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-06-07 US disclosed
EP-0563916-A1 (1H-Indol-1-yl)-2-(amino)acetamides and related (1H-indol-1-yl)-(aminoalkyl)amides, intermediates and a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-10-06 EP disclosed