SCHEMBL8844262

SCHEMBL8844262

CC(C)(C)N(Cc1cccc(C2CCN(Cc3ccccc3)C2)c1)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.51
OPRM1 P35372 1/20 0.47
CHRM2 P08172 1/20 0.46
CHRM3 P20309 1/20 0.46
CHRM4 P08173 2/20 0.44
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
HTT P42858 1/20 0.44
KMT2A Q03164 1/20 0.44
ACHE P22303 1/20 0.43
UBE2M P61081 1/20 0.43
DCUN1D1 Q96GG9 1/20 0.43
MAOB P27338 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8844605 0.90 OPRM1 (0.50) OPRM1CHRM2CHRM3CHRM4KDM4E
SCHEMBL8844223 0.81 DRD2 (0.56) DRD2OPRM1MEN1KMT2AACHE
SCHEMBL22634069 0.78 HTR2C (0.46) MEN1HTTKMT2ADCUN1D1
SCHEMBL4397749 0.77 ACHE (0.53) OPRM1CHRM2CHRM3ACHE
SCHEMBL3524495 0.77 ACHE (0.53) OPRM1CHRM2CHRM3ACHE
SCHEMBL8844412 0.76 JAK3 (0.42) MEN1HTTKMT2A
SCHEMBL9542849 0.76 ROCK2 (0.49) DRD2CHRM4KMT2A
SCHEMBL8844218 0.75 DRD2 (0.60) DRD2MEN1KMT2AACHE
SCHEMBL9482766 0.75 DRD2 (0.54) DRD2CHRM4MEN1KMT2A
SCHEMBL3548653 0.74 OPRM1 (0.47) OPRM1CHRM2CHRM3KDM4EACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5622966-A BACTERICIDES TREATING INFECTIONS WARNER-LAMBERT COMPANY (US) 1997-04-22 US disclosed
US-5446044-A Bactericides WARNER-LAMBERT COMPANY (US) 1995-08-29 US disclosed
US-5384407-A Pyrrolidine compounds WARNER-LAMBERT COMPANY (US) 1995-01-24 US disclosed
US-5342844-A 7-substituted quinolones and naphthyridones as antibacterial agents WARNER-LAMBERT COMPANY (US) 1994-08-30 US disclosed
WO-1993016077-A1 7-SUBSTITUTED QUINOLONES AND NAPHTHYRIDONES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1993-08-19 WO disclosed
US-5221676-A 7-substituted quinolones and naphthyridones as antibacterial agents WARNER-LAMBERT COMPANY (US) 1993-06-22 US disclosed