SCHEMBL8855166

SCHEMBL8855166

COc1cc(C(C)C)c(OC)c2c1C1(C)CCC(=O)C(C)=C1CC2

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.33
CYP3A4 P08684 1/20 0.33
KDM4E B2RXH2 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8855169 0.81
SCHEMBL8855161 0.78
SCHEMBL8855147 0.72 SRD5A1 (0.32)
SCHEMBL8855342 0.71 ALDH1A1 (0.61) ALDH1A1CYP3A4KDM4EHPGD
SCHEMBL8855272 0.67 MAPT (0.37) ALDH1A1CYP3A4
SCHEMBL8855240 0.66 LMNA (0.37) ALDH1A1KDM4EHPGD
SCHEMBL8855310 0.65 CYP3A4 (0.33) ALDH1A1CYP3A4
SCHEMBL9355660 0.64 CYP3A4 (0.33) ALDH1A1CYP3A4KDM4EHPGD
SCHEMBL8855233 0.64 ALDH1A1 (0.35) ALDH1A1KDM4EHPGD
SCHEMBL9360485 0.63 LPAR1 (0.33) ALDH1A1CYP3A4KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-6263688-A None JP disclosed
US-5654343-A NITRIC OXIDE SYNTHESIS INHIBITOR; TREATING ENDOTOXIC SHOCK OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-08-05 US disclosed
EP-0676196-A1 NITROGEN MONOXIDE SYNTHESIS INHIBITOR OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-10-11 EP disclosed
JP-H06263688-A PHENANTHRENE DERIVATIVE OTSUKA PHARMACEUT FACTORY INC 1994-09-20 JP disclosed