SCHEMBL8856166

SCHEMBL8856166

CSc1nc(C)nc(SC)c1NC(=O)N(Cc1ccc(CC(C)(C)C)cc1)C1CCCCCC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
GCGR P47871 2/20 0.36
GIPR P48546 1/20 0.36
ALDH1A1 P00352 4/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
UBE2M P61081 7/20 0.35
DCUN1D1 Q96GG9 7/20 0.35
KDM4E B2RXH2 3/20 0.35
NPC1 O15118 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8856425 0.88 GCGR (0.37) TP53SMN1; SMN2GCGRGIPRALDH1A1
SCHEMBL8856113 0.85 UBE2M (0.40) SMN1; SMN2ALDH1A1UBE2MDCUN1D1
SCHEMBL8817855 0.84 ALDH1A1 (0.44) TP53ALDH1A1ALOX15TSHRHSD17B10
SCHEMBL9056568 0.84 KMT2A (0.41) TP53SMN1; SMN2ALDH1A1ALOX15TSHR
SCHEMBL8808308 0.75 ROCK2 (0.40) TP53SMN1; SMN2ALDH1A1HSD17B10UBE2M
SCHEMBL8344843 0.75 KDM4E (0.42) TP53SMN1; SMN2ALDH1A1HSD17B10UBE2M
SCHEMBL8856219 0.73 UBE2M (0.39) UBE2MDCUN1D1KDM4ECYP1A2CYP3A4
SCHEMBL8808860 0.73 USP2 (0.43) TP53ALDH1A1HSD17B10UBE2MDCUN1D1
SCHEMBL8341852 0.73 UBE2M (0.42) GCGRALDH1A1UBE2MDCUN1D1KDM4E
SCHEMBL8338160 0.73 SLC6A2 (0.44) SMN1; SMN2ALDH1A1UBE2MDCUN1D1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5656634-A N-aryl and N-heteroarylamide and urea derivatives as inhibitors of acyl coenzyme A: cholesterol acyl transferase (ACAT) PFIZER INC. (US) 1997-08-12 US disclosed
US-5362878-A Intermediates for making N-aryl and N-heteroarylamide and urea derivatives as inhibitors of acyl coenzyme A: cholesterol acyl transferase (ACAT) PFIZER INC. (US) 1994-11-08 US disclosed