SCHEMBL8860253

SCHEMBL8860253

Cc1ccc2c(c1)N(Nc1ccncc1)C(=O)C2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP6 P55212 1/20 0.38
CHRM2 P08172 3/20 0.37
CHRM4 P08173 3/20 0.37
CHRM5 P08912 3/20 0.37
CHRM1 P11229 3/20 0.37
CHRM3 P20309 3/20 0.37
HSD17B10 Q99714 1/20 0.36
KMT2A Q03164 4/20 0.36
PKM P14618 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ALDH1A1 P00352 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
MEN1 O00255 2/20 0.34
SLC6A2 P23975 1/20 0.34
NT5E P21589 1/20 0.34
PDE5A O76074 1/20 0.34
RECQL P46063 1/20 0.34
CYP19A1 P11511 2/20 0.33
CYP11B2 P19099 2/20 0.33
AADAT Q8N5Z0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7487924 0.84 CASP6 (0.51) CASP6KMT2APKMSMN1; SMN2ALDH1A1
SCHEMBL8860183 0.80 CASP6 (0.51) CASP6SLC6A2CYP19A1HPGD
SCHEMBL8860233 0.75 CYP19A1 (0.43) KMT2ASMN1; SMN2ALDH1A1MEN1CYP19A1
SCHEMBL7486935 0.70 CASP6 (0.51) CASP6CYP19A1
SCHEMBL7479829 0.70 CASP6 (0.51) CASP6KMT2AMEN1
SCHEMBL7476799 0.70 ALDH1A1 (0.51) CASP6KMT2ASMN1; SMN2ALDH1A1MEN1
SCHEMBL5986263 0.69 HSD17B10 (0.47) CASP6CHRM2CHRM4CHRM5CHRM1
Hydrochloric Acid SCHEMBL8418434 0.69 ALDH1A1 (0.49) CASP6KMT2ASMN1; SMN2ALDH1A1MEN1
Hydrochloric Acid SCHEMBL8418433 0.69 ALDH1A1 (0.49) CASP6KMT2ASMN1; SMN2ALDH1A1MEN1
Hydrochloric Acid SCHEMBL7482266 0.68 ALDH1A1 (0.48) CASP6KMT2ASMN1; SMN2ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686626-A COGNITION ACTIVATORS HOECHST MARION ROUSSEL, INC. (US) 1997-11-11 US disclosed
US-5621116-A CHEMICAL INTERMEDIATES; MEMORY ENHANCERS FOR TREATMENT OF ALZHEIMER*S, ANALGESICS, ANTICONVULSANTS HOECHST MARION ROUSSEL, INC. (US) 1997-04-15 US disclosed
US-5464846-A Learning enhancement, Alzheimer's disease HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1995-11-07 US disclosed
EP-0415102-B1 1,3-Dihydro-1-(pyridinylamino)-2H-indol-2-ones, a process for their preparation and their use as medicaments HOECHST ROUSSEL PHARMA (US) 1995-02-01 EP disclosed
US-5179119-A Cognition activators; alzheimer*s disease HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-01-12 US disclosed
US-5053511-A Analgesics; anticonvulsants; treatment for alzheimers disease HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-10-01 US disclosed
US-5006537-A Analgesics, memory enhancement, Alzheimer* disease HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-04-09 US disclosed
EP-0415102-A1 1,3-Dihydro-1-(pyridinylamino)-2H-indol-2-ones, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-03-06 EP disclosed