SCHEMBL8864841

SCHEMBL8864841

c1ccc(C2N=C3CCCCN3Cc3ccccc32)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 9/20 0.52
BCHE P06276 1/20 0.47
LMNA P02545 2/20 0.46
MEN1 O00255 1/20 0.46
USP2 O75604 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP3A4 P08684 1/20 0.46
KMT2A Q03164 1/20 0.46
KCNH2 Q12809 2/20 0.45
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
SLC6A3 Q01959 2/20 0.37
PRCP P42785 1/20 0.37
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
CHRM3 P20309 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8864671 0.96 ACHE (0.51) ACHEBCHELMNAMEN1USP2
SCHEMBL8556167 0.76 KCNH2 (0.56) LMNAKCNH2SLC6A2SLC6A4SLC6A3
SCHEMBL10377977 0.71 ALPL (0.50) ACHEBCHELMNAALDH1A1KCNH2
SCHEMBL10455191 0.70 NOS1 (0.49) ACHELMNAUSP2ALDH1A1KCNH2
SCHEMBL9540233 0.68 ACHE (1.00) ACHEBCHELMNAMEN1USP2
SCHEMBL10376372 0.66 ALPL (0.51) ACHEBCHELMNAMEN1USP2
SCHEMBL9627472 0.66 SLC6A2 (0.47) MEN1CYP3A4KMT2ASLC6A2SLC6A4
SCHEMBL809711 0.65 NOS1 (0.46) ACHEBCHELMNAMEN1USP2
SCHEMBL8864707 0.65 PRCP (0.46) ACHEKCNH2SLC6A2SLC6A4SLC6A3
SCHEMBL8555627 0.65 KCNH2 (0.72) LMNAKCNH2SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5624922-A Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1997-04-29 US disclosed
US-5380721-A Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1995-01-10 US disclosed