SCHEMBL8865254

SCHEMBL8865254

OC1Cc2ccccc2C1c1c[nH]cn1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 8/20 0.36
P2RX7 Q99572 1/20 0.35
ANPEP P15144 1/20 0.34
OPRK1 P41145 2/20 0.33
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33
GRIN2B Q13224 1/20 0.33
GRIN2C Q14957 1/20 0.33
GRIN3A Q8TCU5 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNA4 P43681 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28513726 0.78 OPRM1 (0.36) OPRM1OPRK1GRIN2DGRIN3BGRIN1
SCHEMBL28478349 0.78 OPRM1 (0.36) OPRM1OPRK1
Hydrochloric Acid SCHEMBL28508991 0.77 OPRM1 (0.35) OPRM1OPRK1
SCHEMBL5827252 0.72 ADRA1A (0.44) P2RX7CHRNB2CHRNA4
SCHEMBL6250927 0.71 ADRA1A (0.54) OPRM1
Hydrochloric Acid SCHEMBL8614363 0.70 ADRA1A (0.43) P2RX7ANPEPCHRNB2CHRNA4
SCHEMBL9354789 0.69 F2R (0.33) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL769063 0.68 ADRA1A (0.55) OPRM1
SCHEMBL3234004 0.67 OPRM1 (0.49) OPRM1ANPEPOPRK1GRIN2DGRIN3B
SCHEMBL16691788 0.67 OPRM1 (0.34) OPRM1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5658938-A HYPOTENSIVE AGENT, ANTIISCHMIC AGENTS U C B S.A. (BE) 1997-08-19 US disclosed
EP-0717037-A1 Substituted 1H-imidazoles having alpha 2-agonistic and alpha 1-antagonistic activity U C B, S.A. (BE) 1996-06-19 EP disclosed