SCHEMBL8865286

SCHEMBL8865286

Cc1cccc(CCCC(O)c2cn(C(c3ccccc3)(c3ccccc3)c3ccccc3)cn2)c1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 7/20 0.39
TAAR1 Q96RJ0 2/20 0.39
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
ASAH1 Q13510 1/20 0.34
CHRM2 P08172 1/20 0.33
CHRM3 P20309 1/20 0.33
CYP19A1 P11511 1/20 0.33
NAAA Q02083 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8865638 0.89 FAAH (0.38) SIRT2CYP11B1CYP11B2
SCHEMBL8865728 0.87 KMT2A (0.38) SIRT2TAAR1ALDH1A1CHRM2CHRM3
SCHEMBL8865570 0.86 SIGMAR1 (0.42) SIRT2TAAR1CHRM2CHRM3
SCHEMBL8986522 0.85 SIRT2 (0.40) SIRT2ALDH1A1KDM4E
SCHEMBL8865406 0.82 ADRB2 (0.43) ALDH1A1KDM4E
SCHEMBL8865969 0.81 SIRT2 (0.34) SIRT2TAAR1CYP11B1CYP11B2CYP19A1
SCHEMBL9518110 0.80 FLT3 (0.39) SIRT2ALDH1A1KDM4ECYP11B1CYP11B2
SCHEMBL10457235 0.79 SIRT2 (0.37) SIRT2CYP11B1CYP11B2
SCHEMBL1736246 0.77 CYP11B1 (0.37) SIRT2CYP11B1CYP11B2
SCHEMBL8865051 0.76 ADRB2 (0.37) SIRT2TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5658938-A HYPOTENSIVE AGENT, ANTIISCHMIC AGENTS U C B S.A. (BE) 1997-08-19 US disclosed
EP-0717037-A1 Substituted 1H-imidazoles having alpha 2-agonistic and alpha 1-antagonistic activity U C B, S.A. (BE) 1996-06-19 EP disclosed