SCHEMBL8865634

SCHEMBL8865634

COc1ccc(Cl)c(CCCC(O)c2cn(C(c3ccccc3)(c3ccccc3)c3ccccc3)cn2)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.35
SLC6A4 P31645 1/20 0.35
SIRT2 Q8IXJ6 12/20 0.35
ACSS2 Q9NR19 2/20 0.33
CASR P41180 2/20 0.33
SLC16A3 O15427 1/20 0.33
SLC16A1 P53985 1/20 0.33
CTSD P07339 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
SLC6A2 P23975 1/20 0.32
HRH2 P25021 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HRH1 P35367 1/20 0.32
OPRM1 P35372 1/20 0.32
DRD3 P35462 1/20 0.32
OPRK1 P41145 1/20 0.32
HTR2B P41595 1/20 0.32
HTR5A P47898 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8865570 0.83 SIGMAR1 (0.42) HTR1ASIRT2SIGMAR1
SCHEMBL8865051 0.82 ADRB2 (0.37) SIRT2SIGMAR1
SCHEMBL8865222 0.78 ABCB1 (0.38) SIRT2
SCHEMBL8865969 0.78 SIRT2 (0.34) SIRT2
SCHEMBL8865406 0.77 ADRB2 (0.43) DRD3TMEM97SIGMAR1
SCHEMBL8865638 0.77 FAAH (0.38) SIRT2
SCHEMBL8865728 0.76 KMT2A (0.38) SIRT2
SCHEMBL9518110 0.75 FLT3 (0.39) SIRT2
SCHEMBL10457235 0.74 SIRT2 (0.37) SIRT2
SCHEMBL8986522 0.74 SIRT2 (0.40) SIRT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5658938-A HYPOTENSIVE AGENT, ANTIISCHMIC AGENTS U C B S.A. (BE) 1997-08-19 US disclosed
EP-0717037-A1 Substituted 1H-imidazoles having alpha 2-agonistic and alpha 1-antagonistic activity U C B, S.A. (BE) 1996-06-19 EP disclosed