SCHEMBL8870542

SCHEMBL8870542

Nc1cc(F)c(F)c(F)c1O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
CA1 P00915 3/20 0.36
CA2 P00918 3/20 0.36
LMNA P02545 2/20 0.36
CA12 O43570 2/20 0.36
CA7 P43166 2/20 0.36
KDM4E B2RXH2 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
CA13 Q8N1Q1 1/20 0.36
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
HSD17B1 P14061 5/20 0.32
HSD17B2 P37059 5/20 0.32
CA4 P22748 2/20 0.31
CA6 P23280 1/20 0.31
CA5A P35218 1/20 0.31
CA9 Q16790 1/20 0.31
CA14 Q9ULX7 1/20 0.31
CA5B Q9Y2D0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11589756 0.81 HSD17B1 (0.39) ALDH1A1CA1CA2LMNACA12
SCHEMBL31150397 0.81 HSD17B1 (0.39) ALDH1A1CA1CA2LMNACA12
SCHEMBL3790406 0.79 VRK1 (0.34) ALDH1A1LMNAKDM4EGAAMAPT
SCHEMBL11796078 0.78 ALDH1A1 (0.41) ALDH1A1LMNAKDM4EGAAMAPT
SCHEMBL3005284 0.75 ALDH1A1 (0.48) ALDH1A1CA1CA2LMNAKDM4E
SCHEMBL5509678 0.75 CES2 (0.38) CA1CA2CA12CA7KDM4E
SCHEMBL2396959 0.75 CA1 (0.40) CA1CA2CA12CA7CA13
SCHEMBL998262 0.75 ALDH1A1 (0.38) ALDH1A1CA1CA2LMNACA12
SCHEMBL30367972 0.75 CA1 (0.40) CA1CA2CA12CA7CA13
SCHEMBL78211 0.74 CA1 (0.43) CA1CA2CA12CA7CA13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5624924-A Quinobenzothiazine antineoplastic agents ABBOTT LABORATORIES (US) 1997-04-29 US disclosed
EP-0608215-A1 QUINOBENZOXAZINE, QUINOBENZOTHIAZINE, AND PYRIDO-ACRIDINE ANTINEOPLASTIC AGENTS ABBOTT LABORATORIES (US) 1994-08-03 EP disclosed
US-5318965-A Administering to treat leukemia, melanoma, carcinoma of lung, colon, ovaries ABBOTT LABORATORIES (US) 1994-06-07 US disclosed
EP-0608215-A4 QUINOBENZOXAZINE, QUINOBENZOTHIAZINE, AND PYRIDO-ACRIDINE ANTINEOPLASTIC AGENTS. ABBOTT LAB (US) 1993-11-11 EP disclosed
WO-1993016702-A1 QUINOBENZOXAZINE, QUINOBENZOTHIAZINE, AND PYRIDO-ACRIDINE ANTINEOPLASTIC AGENTS ABBOTT LABORATORIES (US) 1993-09-02 WO disclosed
WO-1992003136-A1 QUINOBENZOXAZINE, QUINOBENZOTHIAZINE, AND PYRIDO-ACRIDINE ANTINEOPLASTIC AGENTS ABBOTT LABORATORIES (US) 1992-03-05 WO disclosed