SCHEMBL8873046

SCHEMBL8873046

O=C(Nc1ccncn1)C1=C(O)CCc2c1nc1ccccn21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.41
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41
CHRNA4 P43681 1/20 0.41
NAMPT P43490 1/20 0.40
NTRK1 P04629 3/20 0.37
NPC1 O15118 1/20 0.36
TP53 P04637 1/20 0.36
RAB9A P51151 1/20 0.36
CSNK1D P48730 2/20 0.36
CSNK1E P49674 2/20 0.36
ATR Q13535 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
PKM P14618 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MAPT P10636 1/20 0.35
POLB P06746 1/20 0.35
GABRD O14764 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7418872 0.89 NPC1 (0.42) NTRK1NPC1TP53RAB9ACSNK1D
SCHEMBL7958240 0.86 IKBKE (0.41) NTRK1NPC1RAB9AKDM4EMAPT
SCHEMBL7964322 0.85 NTRK1 (0.43) NTRK1NPC1RAB9AKDM4EALDH1A1
SCHEMBL7418952 0.82 RAB9A (0.44) NTRK1NPC1RAB9A
SCHEMBL7420930 0.82 NTRK1 (0.39) NTRK1NPC1RAB9AKDM4EALDH1A1
SCHEMBL7960418 0.81 NTRK1 (0.37) NTRK1NPC1RAB9AKDM4EALDH1A1
SCHEMBL7949796 0.81 RAB9A (0.44) NAMPTNPC1RAB9AKDM4EALDH1A1
SCHEMBL7411535 0.81 SMN1; SMN2 (0.55) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL7420377 0.81 EPHB3 (0.44) NTRK1NPC1RAB9AKDM4EMAPT
SCHEMBL7964531 0.81 CSNK1D (0.40) CSNK1DCSNK1EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5639760-A USEFUL AS MUSCLE RELAXANTS, SEDATIVES, ANXIOLYTICS, ANTICONVULSANTS, AND ANTIDOTES FOR DRUG OVERDOSE MARYANOFF BRUCE E (US) 1997-06-17 US claimed
US-5639760-A USEFUL AS MUSCLE RELAXANTS, SEDATIVES, ANXIOLYTICS, ANTICONVULSANTS, AND ANTIDOTES FOR DRUG OVERDOSE MARYANOFF BRUCE E (US) 1997-06-17 US disclosed