SCHEMBL7960418

SCHEMBL7960418

O=C(Nc1ncc[nH]1)C1=C(O)CCc2c1nc1ccccn21

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 5/20 0.37
KDM4E B2RXH2 3/20 0.35
HSD17B10 Q99714 2/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 2/20 0.35
PKM P14618 1/20 0.35
MAPT P10636 1/20 0.35
POLB P06746 1/20 0.35
KMT2A Q03164 1/20 0.34
NR3C1 P04150 1/20 0.34
RPS6KA3 P51812 1/20 0.34
RPS6KA2 Q15349 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RAB9A P51151 2/20 0.34
NPC1 O15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7964322 0.85 NTRK1 (0.43) NTRK1KDM4EHSD17B10ALDH1A1HPGD
SCHEMBL7418872 0.83 NPC1 (0.42) NTRK1KDM4EALDH1A1PKMKMT2A
SCHEMBL7418952 0.82 RAB9A (0.44) NTRK1KMT2ARAB9ANPC1
SCHEMBL7958240 0.82 IKBKE (0.41) NTRK1KDM4EMAPTKMT2ARAB9A
SCHEMBL8873046 0.81 CHRNB2 (0.41) NTRK1KDM4EHSD17B10ALDH1A1HPGD
SCHEMBL7959855 0.81 LMNA (0.44) NTRK1HPGDMAPTPOLBKMT2A
SCHEMBL7964540 0.80 NPC1 (0.51) KDM4EALDH1A1HPGDPKMMAPT
SCHEMBL7961368 0.80 NTRK1 (0.39) NTRK1KDM4EHSD17B10ALDH1A1HPGD
SCHEMBL7949786 0.80 NTRK1 (0.46) NTRK1KDM4EHSD17B10ALDH1A1HPGD
SCHEMBL7420930 0.80 NTRK1 (0.39) NTRK1KDM4EHSD17B10ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5639760-A USEFUL AS MUSCLE RELAXANTS, SEDATIVES, ANXIOLYTICS, ANTICONVULSANTS, AND ANTIDOTES FOR DRUG OVERDOSE MARYANOFF BRUCE E (US) 1997-06-17 US claimed
US-6218384-B1 FOR THERAPY OF ANXIETY, MUSCLE SPASMS, SLEEPLESSNESS, CONVULSIONS AND BENZODIAZEPINE OVERDOSES ORTHO-MCNEIL PHARMACEUTICAL, INC. 2001-04-17 US disclosed
US-5639760-A USEFUL AS MUSCLE RELAXANTS, SEDATIVES, ANXIOLYTICS, ANTICONVULSANTS, AND ANTIDOTES FOR DRUG OVERDOSE MARYANOFF BRUCE E (US) 1997-06-17 US disclosed