SCHEMBL8876044

SCHEMBL8876044

CCc1c(C(=O)c2ccccc2)oc2c(C(=O)OC)cccc12

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.42
THRB P10828 3/20 0.42
RXFP1 Q9HBX9 2/20 0.41
SLC6A3 Q01959 1/20 0.41
KMT2A Q03164 4/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 1/20 0.40
TSHR P16473 2/20 0.40
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TP53 P04637 1/20 0.38
NR4A2 P43354 1/20 0.38
CYP2C9 P11712 1/20 0.37
BRD4 O60885 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8875450 0.89 CDC25B (0.48) MAPTNPC1TSHRALDH1A1KDM4E
SCHEMBL8877391 0.87 AKR1C3 (0.42) MAPTTHRBRXFP1KMT2ANPC1
SCHEMBL8876122 0.78 MTNR1A (0.43) MAPTKMT2ANPC1RAB9ATSHR
SCHEMBL10550378 0.77 CYP2C19 (0.48) MAPTTHRBSLC6A3KMT2ANPC1
SCHEMBL68630 0.73 LMNA (0.50) MAPTKMT2ATSHRALDH1A1KDM4E
SCHEMBL28434302 0.73 SLC6A3 (0.49) MAPTSLC6A3KMT2ATSHRALDH1A1
SCHEMBL28551648 0.72 TSHR (0.50) MAPTSLC6A3KMT2ATSHRALDH1A1
Aniline SCHEMBL3829674 0.71 ALDH1A1 (0.51) MAPTSLC6A3KMT2ATSHRALDH1A1
SCHEMBL8755551 0.70 TSHR (0.61) MAPTTHRBSLC6A3KMT2ARAB9A
SCHEMBL22481057 0.70 LMNA (0.53) MAPTSLC6A3KMT2ATSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5605896-A Bicyclic heterocyclic derivatives having α1 adrenergic and 5HT1A activities RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1997-02-25 US disclosed