SCHEMBL8879166

SCHEMBL8879166

O=C(Nc1ccc(Cl)c(Cl)c1)NS(=O)(=O)c1ccc2c(c1)CCC2

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA1 Q09470 6/20 0.56
KCNAB1 Q14722 6/20 0.56
CA2 P00918 2/20 0.55
CA9 Q16790 2/20 0.55
CA12 O43570 1/20 0.55
CA1 P00915 1/20 0.55
RAB9A P51151 6/20 0.51
NPC1 O15118 5/20 0.51
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
MAPT P10636 3/20 0.51
EPHX1 P07099 1/20 0.50
EPHX2 P34913 1/20 0.50
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
CASP3 P42574 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
SENP8 Q96LD8 1/20 0.47
SENP7 Q9BQF6 1/20 0.47
SENP6 Q9GZR1 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sulofenur SCHEMBL29359159 0.88 KCNA1 (0.65) KCNA1KCNAB1CA2CA9CA12
Sulofenur SCHEMBL4174 0.88 KCNA1 (0.65) KCNA1KCNAB1CA2CA9CA12
SCHEMBL8878995 0.85 KCNA1 (0.65) KCNA1KCNAB1CA2CA9CA12
SCHEMBL13355422 0.83 RAB9A (0.70) CA2CA9CA12CA1RAB9A
SCHEMBL28766991 0.82 NPC1 (0.67) KCNA1KCNAB1CA2CA9CA12
SCHEMBL15865553 0.82 RAB9A (0.67) KCNA1KCNAB1CA2CA9CA12
Ly-295501 SCHEMBL30351 0.81 PKM (0.58) KCNA1KCNAB1CA2CA9CA12
Ly-295501 SCHEMBL29375534 0.81 PKM (0.58) KCNA1KCNAB1CA2CA9CA12
SCHEMBL8761148 0.81 PKM (0.51) KCNA1KCNAB1CA2CA9CA1
SCHEMBL9486556 0.80 MEN1 (0.67) KCNA1KCNAB1CA2CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5594028-A SULFONYLUREAS ELI LILLY AND COMPANY (US) 1997-01-14 US disclosed
US-5116874-A Aminocarbonyl sulfonamide derivatives ELI LILLY AND COMPANY (US) 1992-05-26 US disclosed
EP-0222475-B1 SULFONYL UREAS WITH ANTI-TUMOUR ACTIVITY ELI LILLY AND COMPANY (US) 1989-11-29 EP disclosed
EP-0222475-A1 Sulfonyl ureas with anti-tumour activity ELI LILLY AND COMPANY (US) 1987-05-20 EP disclosed