Ly-295501

Ly-295501

SCHEMBL30351

O=C(Nc1ccc(Cl)c(Cl)c1)NS(=O)(=O)c1ccc2c(c1)CCO2

nearest known ligand 0.58

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 3/20 0.58
MAPT P10636 2/20 0.58
IDH1 O75874 1/20 0.52
CA2 P00918 3/20 0.50
CA9 Q16790 3/20 0.50
CA1 P00915 2/20 0.50
PKLR P30613 1/20 0.50
CA12 O43570 1/20 0.50
HDAC3 O15379 1/20 0.48
HDAC4 P56524 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC10 Q969S8 1/20 0.48
HDAC11 Q96DB2 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
HDAC9 Q9UKV0 1/20 0.48
HDAC5 Q9UQL6 1/20 0.48
MAOB P27338 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ly-295501 SCHEMBL29375534 1.00 PKM (0.58) PKMMAPTIDH1CA2CA9
SCHEMBL15865555 0.90 IDH1 (0.59) PKMMAPTIDH1CA2CA9
SCHEMBL8877626 0.89 PKM (0.70) PKMMAPTIDH1CA2CA9
SCHEMBL8879166 0.81 KCNA1 (0.56) MAPTCA2CA9CA1CA12
SCHEMBL6425171 0.81 PKM (0.53) PKMMAPTIDH1PKLRHDAC3
SCHEMBL8761148 0.78 PKM (0.51) PKMMAPTCA2CA9CA1
SCHEMBL5779906 0.77 CCR2 (0.69) PKMMAPTIDH1CA2CA9
SCHEMBL9486556 0.77 MEN1 (0.67) MAPTCA2CA9CA1CA12
SCHEMBL9476125 0.76 EPHX1 (0.47) MAPTCA2CA9CA1CA12
SCHEMBL7993384 0.76 KCNA1 (0.51) PKMMAPTEPHX1EPHX2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1639 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2805945-B1 Amide substituted indazoles as poly(ADP-ribose)polymerase (PARP) inhibitors MSD ITALIA SRL (IT) 2019-04-03 EP claimed
US-20140301976-A1 NOVEL HYDROXAMATES AS THERAPEUTIC AGENTS PHARMACYCLICS, INC. 2014-10-09 US claimed
US-8779171-B2 Hydroxamates as therapeutic agents PHARMACYCLICS, INC. (US) 2014-07-15 US claimed
US-20130142758-A1 NOVEL HYDROXAMATES AS THERAPEUTIC AGENTS PHARMACYCLICS, INC. (US) 2013-06-06 US claimed
US-20100291592-A1 NOVEL MARKER FOR SENSITIVITY AGAINST SULFONAMIDE COMPOUND EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-11-18 US claimed
US-20090047365-A1 Novel Concomitant Use of Sulfonamide Compound with Anti-Cancer Agent EISAI R & D MANAGEMENT CO., LTD. (JP) 2009-02-19 US claimed
US-20090047278-A1 Novel Combinational Use of Sulfonamide Compound EISAI R & D MANAGEMENT CO., LTD. (JP) 2009-02-19 US claimed
EP-2015070-A1 NOVEL MARKER FOR SENSITIVITY AGAINST SULFONAMIDE COMPOUND Eisai R&D Management Co., Ltd. (JP) 2009-01-14 EP claimed
US-20080286282-A1 Novel Use of Sulfonamide Compound in Combination with Angiogenesis Inhibitor EISAI R & D MANAGEMENT CO., LTD. (JP) 2008-11-20 US claimed
EP-1862179-A1 NOVEL USE OF SULFONAMIDE COMPOUND IN COMBINATION WITH ANGIOGENESIS INHIBITOR Eisai R&D Management Co., Ltd. (JP) 2007-12-05 EP claimed
EP-1859793-A1 NOVEL COMBINATIONAL USE OF SULFONAMIDE COMPOUND Eisai R&D Management Co., Ltd. (JP) 2007-11-28 EP claimed
EP-1859797-A1 NOVEL CONCOMITANT USE OF SULFONAMIDE COMPOUND WITH ANTI-CANCER AGENT Eisai R&D Management Co., Ltd. (JP) 2007-11-28 EP claimed
EP-1797877-A1 JOINT USE OF SULFONAMIDE BASED COMPOUND WITH ANGIOGENESIS INHIBITOR Eisai Co., Ltd. (JP) 2007-06-20 EP claimed
US-20060135486-A1 Use of sulfonamide-including compounds in combination with angiogenesis inhibitors EISAI CO., LTD. (JP) 2006-06-22 US claimed
EP-0583960-B1 Synthesis of bicyclic aromatic sulfonic acids, sulfonyl chlorides and sulfonamides LILLY CO ELI (US) 1997-05-21 EP claimed
EP-0583960-A2 Synthesis of bicyclic aromatic sulfonic acids, sulfonyl chlorides and sulfonamides ELI LILLY AND COMPANY (US) 1994-02-23 EP claimed
US-20260132164-A1 PNU ANTHRACYCLINE DERIVATIVES AND METHODS OF USE THEREOF MERCK SHARP & DOHME LLC (US) 2026-05-14 US disclosed
EP-4076459-B1 PRMT5 INHIBITORS MERCK SHARP & DOHME LLC (US) 2026-04-29 EP disclosed
EP-0555036-A2 Antitumor compositions and methods of treatment ELI LILLY AND COMPANY (US) 1993-08-11 EP disclosed
EP-0555036-A2 Antitumor compositions and methods of treatment ELI LILLY AND COMPANY (US) 1993-08-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090047278-A1 Novel Combinational Use of Sulfonamide Compound EGFR, KIT, ERBB2 PKM 2667/4885MAPT 4340/4885IDH1 3433/4885
US-20060135486-A1 Use of sulfonamide-including compounds in combination with angiogenesis inhibitors FLT4, KDR, FLT1 PKM 3395/4885MAPT 3475/4885IDH1 513/4885
US-20130142758-A1 NOVEL HYDROXAMATES AS THERAPEUTIC AGENTS HDAC1, HDAC3, HDAC5 PKM 3513/4885MAPT 4192/4885IDH1 129/4885
US-20140301976-A1 NOVEL HYDROXAMATES AS THERAPEUTIC AGENTS HDAC1, HDAC3, HDAC5 PKM 3513/4885MAPT 4192/4885IDH1 129/4885
US-20090047365-A1 Novel Concomitant Use of Sulfonamide Compound with Anti-Cancer Agent TOP1, TOP2A, TOP2B PKM 1903/4885MAPT 789/4885IDH1 782/4885
US-20260132164-A1 PNU ANTHRACYCLINE DERIVATIVES AND METHODS OF USE THEREOF TOP1, NCL, NOLC1 PKM 3662/4885MAPT 4774/4885IDH1 122/4885
US-20080286282-A1 Novel Use of Sulfonamide Compound in Combination with Angiogenesis Inhibitor KDR, FLT4, FLT1 PKM 2169/4885MAPT 3691/4885IDH1 1233/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.