SCHEMBL8879639

SCHEMBL8879639

COC(=O)CCc1ccc(CCBr)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 2/20 0.50
CYP4A11 Q02928 2/20 0.50
IDO1 P14902 1/20 0.50
F2RL1 P55085 1/20 0.49
ADRB2 P07550 1/20 0.48
ADRB1 P08588 1/20 0.48
EPHX2 P34913 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46
ALDH1A1 P00352 2/20 0.46
LMNA P02545 1/20 0.46
MAPT P10636 1/20 0.46
HTT P42858 1/20 0.46
KMT2A Q03164 1/20 0.46
HSD17B10 Q99714 1/20 0.46
PTPN1 P18031 1/20 0.45
TSHR P16473 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
CA12 O43570 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22922181 0.90 CYP4F2 (0.59) CYP4F2CYP4A11IDO1F2RL1ADRB2
SCHEMBL27700759 0.89 TSHR (0.48) CYP4F2CYP4A11EPHX2ALDH1A1LMNA
SCHEMBL1483117 0.89 CYP4F2 (0.50) CYP4F2CYP4A11IDO1F2RL1ADRB2
SCHEMBL9670477 0.86 THRA (0.53) CYP4F2CYP4A11IDO1F2RL1ADRB2
SCHEMBL8158284 0.85 CYP4F2 (0.70) CYP4F2CYP4A11ALDH1A1LMNAMAPT
SCHEMBL516422 0.85 IDO1 (0.65) CYP4F2CYP4A11IDO1F2RL1ADRB2
SCHEMBL28549048 0.83 ADRB2 (0.54) F2RL1ADRB2ADRB1ALDH1A1LMNA
SCHEMBL10583619 0.83 TSHR (0.50) CYP4F2CYP4A11F2RL1EPHX2ALDH1A1
Hydrochloric Acid SCHEMBL16062033 0.83 IDO1 (0.63) CYP4F2CYP4A11IDO1F2RL1ADRB2
SCHEMBL1410420 0.82 CYP4A11 (0.56) CYP4F2CYP4A11IDO1F2RL1ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5624948-A TREATMENT OF BRONCHIAL ASTHMA KISSEI PHARMACEUTICAL CO., LTD. (JP) 1997-04-29 US disclosed
EP-0699668-A1 1-(2-BENZIMIDAZOLYL)-1,5-DIAZACYCLOOCTANE DERIVATIVE Kissei Pharmaceutical Co., Ltd. (JP) 1996-03-06 EP disclosed