SCHEMBL28549048

SCHEMBL28549048

COC(=O)CCc1ccc(OCCBr)cc1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.54
ADRB1 P08588 1/20 0.54
LMNA P02545 2/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
LTA4H P09960 2/20 0.50
PPARG P37231 1/20 0.49
KMT2A Q03164 3/20 0.49
FFAR1 O14842 4/20 0.49
F2RL1 P55085 1/20 0.49
ATM Q13315 1/20 0.48
ALDH1A1 P00352 2/20 0.46
MAPT P10636 1/20 0.46
HTT P42858 1/20 0.46
HSD17B10 Q99714 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7037985 0.92 ADRB2 (0.53) ADRB2ADRB1LMNAL3MBTL1LTA4H
SCHEMBL2159817 0.91 LTA4H (0.50) ADRB2ADRB1LMNAL3MBTL1LTA4H
SCHEMBL4944581 0.91 ADRB2 (0.52) ADRB2ADRB1LMNAL3MBTL1LTA4H
SCHEMBL2170785 0.90 FFAR1 (0.50) ADRB2ADRB1LMNAL3MBTL1LTA4H
SCHEMBL7528179 0.86 LMNA (0.62) ADRB2ADRB1LMNAL3MBTL1FFAR1
SCHEMBL1495266 0.84 ADRB2 (0.54) ADRB2ADRB1LMNAL3MBTL1LTA4H
SCHEMBL27545059 0.84 ADRB2 (0.54) ADRB2ADRB1LMNAL3MBTL1LTA4H
SCHEMBL13932451 0.84 FFAR1 (0.60) ADRB2ADRB1LMNAL3MBTL1LTA4H
SCHEMBL28543599 0.84 ADRB2 (0.54) ADRB2ADRB1LMNAL3MBTL1LTA4H
SCHEMBL2437986 0.84 ALDH1A1 (0.54) LMNAL3MBTL1LTA4HKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108239029-B Preparation and medical application of tetrahydroisoquinoline compounds and salts thereof 中国医学科学院药物研究所 2021-04-13 CN disclosed