SCHEMBL8879807

SCHEMBL8879807

O=C(O)CCNC(=O)C12CC3CC(CC(C3)C1)C2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 1.00
HTT P42858 1/20 1.00
KMT2A Q03164 3/20 0.53
MEN1 O00255 2/20 0.53
HPGD P15428 1/20 0.53
EPHX2 P34913 4/20 0.50
ITGB1 P05556 3/20 0.50
ITGA4 P13612 3/20 0.50
HSD11B1 P28845 2/20 0.49
ALOX5 P09917 1/20 0.47
ALDH1A1 P00352 1/20 0.46
CYP17A1 P05093 1/20 0.46
CYP19A1 P11511 1/20 0.46
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16365921 0.86 KDM4E (0.76) KDM4EHTTKMT2AMEN1HPGD
SCHEMBL1758666 0.81 HTT (0.68) KDM4EHTTKMT2AMEN1HPGD
SCHEMBL28334704 0.81 KDM4E (0.68) KDM4EHTTKMT2AMEN1HPGD
SCHEMBL8655345 0.79 KDM4E (0.66) KDM4EHTTKMT2AMEN1HPGD
SCHEMBL13873443 0.79 HTT (0.66) KDM4EHTTKMT2AMEN1HPGD
SCHEMBL7778418 0.78 KDM4E (0.64) KDM4EHTTKMT2AMEN1HPGD
SCHEMBL20999491 0.77 KDM4E (0.63) KDM4EHTTKMT2AMEN1HPGD
SCHEMBL27004615 0.76 HTT (0.62) KDM4EHTTKMT2AMEN1HPGD
SCHEMBL17702625 0.76 KMT2A (0.70) KDM4EHTTKMT2AMEN1HPGD
SCHEMBL22005490 0.76 KDM4E (0.60) KDM4EHTTKMT2AMEN1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5679701-A INHIBITS CALCIUM UPTAKE IN CARDIAC MUSCLE; HAS NEGATIVE INOTROPIC EFFECT ON MAMMALIAN CARDIAC MUSCLE INDIANA UNIVERSITY FOUNDATION (US) 1997-10-21 US disclosed
US-5510500-A RADIO-IODINATED ALANINE DERIVATIVES AS LABELS INDIANA UNIVERSITY FOUNDATION (US) 1996-04-23 US disclosed
US-5432288-A Useful in effecting calcium efflux in tissue INDIANA UNIVERSITY FOUNDATION (US) 1995-07-11 US disclosed
WO-1992018499-A1 NOVEL ESTER DERIVATIVES OF RYANODINE AND DEHYDRORYANODINE INDIANA UNIVERSITY FOUNDATION (US) 1992-10-29 WO disclosed